SCHEMBL12640800

SCHEMBL12640800

COC(=O)c1c(N)nc(N)nc1Nc1cccc(C)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 5/20 0.55
MAPT P10636 5/20 0.55
CISD2 Q8N5K1 1/20 0.47
LMNA P02545 1/20 0.47
TSHR P16473 1/20 0.47
MAPK1 P28482 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.45
EGFR P00533 1/20 0.44
ROCK1 Q13464 1/20 0.44
BRAF P15056 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
NOD1 Q9Y239 1/20 0.43
AURKB Q96GD4 3/20 0.43
SYK P43405 3/20 0.43
ALDH1A1 P00352 1/20 0.43
HPGD P15428 1/20 0.43
HSD17B10 Q99714 1/20 0.43
PRKD3 O94806 1/20 0.42
CSF1R P07333 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12640925 0.81 CISD2 (0.46) TP53MAPTCISD2LMNATSHR
SCHEMBL12640993 0.80 FER (0.52) MAPK1NPC1RAB9AAURKBSYK
SCHEMBL1989865 0.78 NFKB1 (0.51) TP53MAPTCISD2LMNATSHR
SCHEMBL1986001 0.78 NFKB1 (0.51) TP53MAPTCISD2LMNATSHR
SCHEMBL1988610 0.76 LMNA (0.48) TP53MAPTCISD2LMNATSHR
SCHEMBL1986008 0.74 KMT2A (0.46) TP53MAPTCISD2LMNATSHR
SCHEMBL1986224 0.73 FER (0.46) TP53MAPTCISD2LMNATSHR
SCHEMBL16743301 0.72 KDR (0.50) TP53MAPTMAPK1EGFRROCK1
SCHEMBL15887222 0.71 NPC1 (0.50) TP53MAPTLMNATSHRNPC1
SCHEMBL10254010 0.71 NFKB1 (0.49) TP53MAPTLMNATSHRMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011079051-A1 FUSED HETEROAROMATIC PYRROLIDINONES AS SYK INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-06-30 WO disclosed