SCHEMBL1270280

SCHEMBL1270280

CC(c1cc2ccccc2[nH]1)C1C(=O)c2ccccc2OC12CCNCC2

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 8/20 0.37
KCNH2 Q12809 7/20 0.37
CYP2D6 P10635 5/20 0.37
BRD4 O60885 3/20 0.36
CREBBP Q92793 2/20 0.36
ALOX5 P09917 1/20 0.34
MAOB P27338 2/20 0.33
OPRK1 P41145 3/20 0.33
KDR P35968 2/20 0.32
CHEK1 O14757 1/20 0.32
HRH4 Q9H3N8 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
AURKA O14965 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13339981 0.72 OPRD1 (0.43) OPRD1KCNH2CYP2D6OPRK1
Hydrochloric Acid SCHEMBL3495476 0.71 OPRD1 (0.42) OPRD1KCNH2CYP2D6OPRK1
SCHEMBL12480913 0.70 ATM (0.44) OPRD1KCNH2CYP2D6OPRK1
SCHEMBL2589311 0.66 OPRD1 (0.44) OPRD1KCNH2CYP2D6OPRK1
SCHEMBL1269847 0.66 HTT (0.38) OPRD1KCNH2
SCHEMBL12482165 0.65 MAOB (0.46) OPRD1KCNH2CYP2D6MAOBOPRK1
SCHEMBL3457811 0.64 OPRD1 (0.45) OPRD1KCNH2CYP2D6OPRK1
SCHEMBL2591939 0.63 OPRD1 (0.39) OPRD1KCNH2CYP2D6OPRK1
SCHEMBL17276804 0.62 OPRD1 (0.43) OPRD1KCNH2CYP2D6OPRK1
SCHEMBL14972718 0.62 EPHX2 (0.38) OPRD1KCNH2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2279187-A1 SPIROCYCLIC DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS DAC S.r.l. (IT) 2011-02-02 EP claimed
WO-2009127609-A1 SPIROCYCLIC DERIVATIVES AS HISTONE DEACETYLASE INHIBITORS DAC S.R.L. (IT) 2009-10-22 WO claimed