SCHEMBL12716705

SCHEMBL12716705

CC(=O)CC1Cc2cccc([N+](=O)[O-])c2C1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
DRD2 P14416 1/20 0.38
ADRA2C P18825 1/20 0.38
NPY1R P25929 1/20 0.38
NPY5R Q15761 1/20 0.38
ERN1 O75460 1/20 0.38
TSHR P16473 3/20 0.38
TP53 P04637 1/20 0.38
ALOX15 P16050 1/20 0.38
TDP1 Q9NUW8 3/20 0.38
GPR35 Q9HC97 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
TAS1R2 Q8TE23 1/20 0.36
ALDH1A1 P00352 4/20 0.36
MAPT P10636 2/20 0.36
MAPK1 P28482 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2246781 0.82 GPR35 (0.42) CHRNB2CHRNA4DRD2ADRA2CNPY1R
SCHEMBL2242996 0.81 CHRNB2 (0.35) CHRNB2CHRNA4DRD2ADRA2CNPY1R
SCHEMBL12355698 0.80 CHRNB2 (0.40) CHRNB2CHRNA4DRD2ADRA2CNPY1R
SCHEMBL7517485 0.78 TDP1 (0.41) CHRNB2CHRNA4ERN1TSHRALOX15
SCHEMBL1415461 0.78 MTNR1A (0.47) CHRNB2CHRNA4DRD2ADRA2CNPY1R
SCHEMBL1573308 0.75 TDP1 (0.38) CHRNB2CHRNA4ERN1TSHRTDP1
SCHEMBL13332612 0.75 MTNR1A (0.44)
SCHEMBL5916971 0.74 GPR35 (0.46) CHRNB2CHRNA4ERN1TSHRALOX15
SCHEMBL14017372 0.74 TDP1 (0.44) CHRNB2CHRNA4TSHRALOX15TDP1
SCHEMBL1080845 0.74 TDP1 (0.44) CHRNB2CHRNA4TSHRALOX15TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2048132-B1 Tetrahydro-naphthalene and urea derivatives XENTION LTD (GB) 2011-04-13 EP disclosed