SCHEMBL127910

SCHEMBL127910

Cc1ccc(CO)c(Br)c1C

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NCEH1 Q6PIU2 1/20 0.38
PDCD1 Q15116 2/20 0.35
CD274 Q9NZQ7 2/20 0.35
SHBG P04278 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2A6 P11509 1/20 0.32
TSHR P16473 1/20 0.32
GABRA1 P14867 1/20 0.30
GABRB2 P47870 1/20 0.30
TRPA1 O75762 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL287086 0.82 PDCD1 (0.39) NCEH1PDCD1CD274SHBGGABRA1
SCHEMBL31719921 0.78 PDCD1 (0.33) PDCD1CD274
SCHEMBL358606 0.78 PDCD1 (0.43) PDCD1CD274SHBGCYP1A2CYP2A6
SCHEMBL128934 0.77 PON1 (0.40) NCEH1GABRA1GABRB2
SCHEMBL6406593 0.77 NCEH1 (0.34) NCEH1CYP1A2GABRA1GABRB2
Phosphine SCHEMBL3840466 0.76 PDCD1 (0.42) PDCD1CD274SHBGCYP1A2CYP2A6
Ammonia Solution, Strong SCHEMBL439692 0.76 PDCD1 (0.42) PDCD1CD274SHBGCYP1A2CYP2A6
SCHEMBL10557023 0.76 SHBG (0.39) PDCD1CD274SHBG
SCHEMBL128869 0.75 SMN1; SMN2 (0.50) NCEH1CYP1A2TSHR
SCHEMBL205613 0.74 PDCD1 (0.36) PDCD1CD274SHBGCYP1A2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11077090-B2 Compounds and compositions and uses thereof SUNOVION PHARMACEUTICALS INC. (MA) 2021-08-03 US disclosed
EP-3490607-A1 COMPOUNDS AND COMPOSITIONS AND USES THEREOF Sunovion Pharmaceuticals Inc. (US) 2019-06-05 EP disclosed
WO-2018023070-A1 COMPOUNDS AND COMPOSITIONS AND USES THEREOF SUNOVION PHARMACEUTICALS, INC. (US) 2018-02-01 WO disclosed
US-20180028492-A1 COMPOUNDS AND COMPOSITIONS AND USES THEREOF PGI DRUG DISCOVERY LLC 2018-02-01 US disclosed
US-9227966-B2 Antimicrobial agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2016-01-05 US disclosed
US-8933096-B2 Antimicrobial agents Rugers, The State University of New Jersey (US) 2015-01-13 US disclosed
US-20140315939-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-10-23 US disclosed
US-20130116278-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2013-05-09 US disclosed
US-20120059026-A1 ANTIMICROBIAL AGENTS UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 2012-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116278-A1 ANTIMICROBIAL AGENTS MRPL21, ARG1, RPP30 NCEH1 3014/4885PDCD1 4176/4885CD274 3356/4885
US-20120059026-A1 ANTIMICROBIAL AGENTS ZYX, Q6ZSR9, ZC3HAV1L NCEH1 990/4885PDCD1 4544/4885CD274 4209/4885
US-11077090-B2 Compounds and compositions and uses thereof ACHE, CHAT, MAOB NCEH1 456/4885PDCD1 4720/4885CD274 4809/4885
US-20180028492-A1 COMPOUNDS AND COMPOSITIONS AND USES THEREOF ACHE, CHAT, MAOB NCEH1 456/4885PDCD1 4720/4885CD274 4809/4885
US-20140315939-A1 ANTIMICROBIAL AGENTS ZYX, Q6ZSR9, ZC3HAV1L NCEH1 1101/4885PDCD1 4541/4885CD274 4203/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.