SCHEMBL1279944

SCHEMBL1279944

CC1COC(Cn2cncn2)(c2cc(F)c(Oc3ccccc3)c(F)c2)O1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSP90AA1 P07900 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CYP3A4 P08684 13/20 0.41
THRB P10828 1/20 0.41
GAA P10253 1/20 0.40
HSD17B10 Q99714 1/20 0.40
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
TSHR P16473 2/20 0.36
NR1I2 O75469 1/20 0.35
LMNA P02545 1/20 0.35
FYN P06241 1/20 0.35
PGR P06401 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
ADRA2A P08913 1/20 0.35
CHRM1 P11229 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1280255 0.89 HSP90AA1 (0.45) HSP90AA1NPSR1CYP3A4THRBGAA
SCHEMBL9458158 0.86 HSP90AA1 (0.53) HSP90AA1NPSR1CYP3A4THRBGAA
SCHEMBL1279754 0.84 CYP3A4 (0.46) HSP90AA1NPSR1CYP3A4THRBGAA
SCHEMBL1280067 0.83 CYP3A4 (0.44) HSP90AA1NPSR1CYP3A4THRBGAA
SCHEMBL28608936 0.82 HSP90AA1 (0.57) HSP90AA1NPSR1CYP3A4THRBGAA
SCHEMBL28602335 0.82 HSP90AA1 (0.57) HSP90AA1NPSR1CYP3A4THRBGAA
SCHEMBL11544305 0.82 HSP90AA1 (0.57) HSP90AA1NPSR1CYP3A4THRBGAA
SCHEMBL1280620 0.82 HSP90AA1 (0.46) HSP90AA1NPSR1CYP3A4THRBGAA
SCHEMBL1279580 0.81
SCHEMBL1279774 0.81 CYP3A4 (0.47) HSP90AA1NPSR1CYP3A4THRBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102459241-A Triazole compounds with sulfur substituents BASF SE 2012-05-16 CN disclosed
EP-2443109-A1 TRIAZOLE COMPOUNDS CARRYING A SULFUR SUBSTITUENT BASF SE (DE) 2012-04-25 EP disclosed
US-20120088663-A1 Triazole Compounds Carrying a Sulfur Substituent BASF SE (DE) 2012-04-12 US disclosed
WO-2010146114-A1 TRIAZOLE COMPOUNDS CARRYING A SULFUR SUBSTITUENT BASF SE (DE) 2010-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120088663-A1 Triazole Compounds Carrying a Sulfur Substituent TST, STS, SQOR HSP90AA1 3133/4885NPSR1 3019/4885CYP3A4 39/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.