SCHEMBL12809583

SCHEMBL12809583

Cn1ncc(C(=O)NC2CCC3CC4CC(C3)C2C4)c1N1CCC(O)C1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.38
LMNA P02545 2/20 0.38
IDH1 O75874 1/20 0.36
HSD11B1 P28845 4/20 0.35
HSD17B10 Q99714 2/20 0.35
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
OPRK1 P41145 2/20 0.33
PIM1 P11309 1/20 0.33
KDM4E B2RXH2 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
JAK2 O60674 1/20 0.32
NTRK1 P04629 1/20 0.32
CNR2 P34972 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12809585 1.00 HTT (0.38) HTTLMNAIDH1HSD11B1HSD17B10
SCHEMBL12809749 0.94 LMNA (0.39) HTTLMNAIDH1HSD11B1HSD17B10
SCHEMBL12809710 0.88 HTT (0.40) HTTLMNAIDH1HSD11B1HSD17B10
SCHEMBL12809574 0.88 HSD11B1 (0.33) LMNAIDH1HSD11B1HSD17B10ALDH1A1
SCHEMBL12809702 0.87 HTT (0.39) HTTLMNAIDH1HSD11B1HSD17B10
SCHEMBL12809582 0.87 HTT (0.39) HTTLMNAIDH1HSD11B1HSD17B10
SCHEMBL12809748 0.87 HRH4 (0.41) HTTLMNAIDH1HSD11B1HSD17B10
SCHEMBL1406964 0.86 LMNA (0.52) HTTLMNAHSD11B1ALDH1A1SMN1; SMN2
SCHEMBL1406813 0.86 LMNA (0.52) HTTLMNAHSD11B1ALDH1A1SMN1; SMN2
SCHEMBL12809575 0.85 IDH1 (0.37) HTTLMNAIDH1HSD11B1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2295411-A1 Pyrazoles as 11-beta-hsd-1 F. Hoffmann-La Roche AG (CH) 2011-03-16 EP disclosed
WO-2007107470-A2 PYRAZOLES AS 11-BETA-HSD-1 F. HOFFMANN-LA ROCHE AG (CH) 2007-09-27 WO disclosed