SCHEMBL12830656

SCHEMBL12830656

COc1cc(C)cc(/C=C/c2ccc([N+](=O)[O-])cc2)c1

nearest known ligand 0.83

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.83
PTGS1 P23219 2/20 0.83
TLR9 Q9NR96 1/20 0.59
CYP19A1 P11511 4/20 0.58
NFE2L2 Q16236 2/20 0.56
MAOA P21397 1/20 0.52
MAOB P27338 1/20 0.52
ESR1 P03372 2/20 0.51
NQO2 P16083 2/20 0.51
ABL1 P00519 1/20 0.51
TTR P02766 1/20 0.51
CYP1A1 P04798 1/20 0.51
CYP1A2 P05177 1/20 0.51
ABCB1 P08183 1/20 0.51
ALOX5 P09917 1/20 0.51
BCR P11274 1/20 0.51
CYP1B1 Q16678 1/20 0.51
TUBB4A P04350 1/20 0.51
TUBB P07437 1/20 0.51
TUBA3C P0DPH7 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3392246 0.91 PTGS2 (1.00) PTGS2PTGS1TLR9CYP19A1NFE2L2
SCHEMBL4735253 0.91 PTGS2 (1.00) PTGS2PTGS1TLR9CYP19A1NFE2L2
SCHEMBL4733440 0.91 PTGS2 (1.00) PTGS2PTGS1TLR9CYP19A1NFE2L2
SCHEMBL3395077 0.84 PTGS2 (0.86) PTGS2PTGS1TLR9CYP19A1NFE2L2
SCHEMBL1005735 0.82 PTGS2 (0.78) PTGS2PTGS1TLR9CYP19A1NFE2L2
SCHEMBL1005734 0.82 PTGS2 (0.78) PTGS2PTGS1TLR9CYP19A1NFE2L2
SCHEMBL12535856 0.81 PTGS2 (0.78) PTGS2PTGS1CYP19A1ESR1NQO2
SCHEMBL10312395 0.81 RELA (0.68) PTGS2PTGS1CYP19A1ESR1NQO2
SCHEMBL1405456 0.81 PTGS2 (0.75) PTGS2PTGS1TLR9CYP19A1NFE2L2
SCHEMBL1405454 0.81 PTGS2 (0.75) PTGS2PTGS1TLR9CYP19A1NFE2L2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2289504-A2 SIRT1 modulators for manipulating cell/organism lifespan/stress response President and Fellows of Harvard College (US) 2011-03-02 EP disclosed