SCHEMBL12832452

SCHEMBL12832452

O=C(O)C1CC(C(=O)c2cccc(C(F)(F)F)c2)C1

nearest known ligand 0.56

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.56
SRD5A2 P31213 1/20 0.51
LMNA P02545 3/20 0.50
HSD11B1 P28845 1/20 0.50
MGLL Q99685 1/20 0.49
NOTUM Q6P988 1/20 0.49
POLB P06746 1/20 0.48
HPGD P15428 1/20 0.48
MEN1 O00255 1/20 0.47
KMT2A Q03164 1/20 0.47
MAOB P27338 1/20 0.47
KCNK3 O14649 1/20 0.47
NPSR1 Q6W5P4 1/20 0.46
P2RX1 P51575 1/20 0.46
S1PR5 Q9H228 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL377011 0.84 CES2 (0.62) CES2SRD5A2LMNAHSD11B1MGLL
SCHEMBL7418491 0.79 HSD11B1 (0.56) CES2SRD5A2LMNAHSD11B1MGLL
Hydrochloric Acid SCHEMBL11517089 0.78 HTR2C (0.56) CES2SRD5A2LMNAHSD11B1MGLL
SCHEMBL7456011 0.77 CES2 (0.53) CES2SRD5A2LMNAHSD11B1MGLL
SCHEMBL1498423 0.75 ELOVL6 (0.53) CES2LMNANOTUMPOLBMEN1
SCHEMBL10476083 0.75 ELOVL6 (0.53) CES2LMNANOTUMPOLBMEN1
SCHEMBL1498422 0.75 ELOVL6 (0.53) CES2LMNANOTUMPOLBMEN1
SCHEMBL4848676 0.75 CES2 (0.89) CES2SRD5A2LMNAPOLBHPGD
SCHEMBL29433907 0.75 SRD5A2 (0.77) CES2SRD5A2LMNAPOLBHPGD
SCHEMBL40186 0.75 SRD5A2 (0.77) CES2SRD5A2LMNAPOLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011035159-A1 ARYL SULPHONE DERIVATIVES AS CALCIUM CHANNEL BLOCKERS ZALICUS PHARMACEUTICALS LTD. (CA) 2011-03-24 WO disclosed