SCHEMBL12833909

SCHEMBL12833909

COc1ncccc1-c1ccc(O)c(-c2nc3cc(C(=O)NC4CCc5cncn5C4)ccc3[nH]2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.37
HDAC1 Q13547 1/20 0.37
HDAC2 Q92769 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
CARM1 Q86X55 2/20 0.36
MAPK14 Q16539 1/20 0.36
SMYD3 Q9H7B4 1/20 0.36
TBK1 Q9UHD2 2/20 0.35
HPSE Q9Y251 1/20 0.35
GSK3B P49841 1/20 0.35
FLT3 P36888 1/20 0.35
CRBN Q96SW2 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
NAMPT P43490 1/20 0.33
PDE10A Q9Y233 1/20 0.33
RIPK1 Q13546 1/20 0.33
KDM4E B2RXH2 1/20 0.33
NPC1 O15118 1/20 0.33
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12834192 0.86 MAPK14 (0.47) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL14090786 0.86 ACSS2 (0.42) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL12833757 0.85 SMN1; SMN2 (0.45) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL12833745 0.84 SMN1; SMN2 (0.47) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL1509532 0.84 CARM1 (0.43) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL12833879 0.82 HDAC6 (0.41) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL12833424 0.82 PDE10A (0.44) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL12834499 0.82 HPGDS (0.43) HDAC3HDAC1HDAC2HDAC8HDAC6
SCHEMBL12833953 0.81 TBK1 (0.46) CARM1TBK1GSK3BSMN1; SMN2
SCHEMBL12833445 0.81 CARM1 (0.47) HDAC3HDAC1HDAC2HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2298770-A1 Heterocyclic compounds as TrkA modulators ChemBridge Corporation (US) 2011-03-23 EP disclosed