SCHEMBL1285396

SCHEMBL1285396

Cc1cc(O)cc(O)c1[N+](=O)[O-]

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.44
ACHE P22303 2/20 0.44
ALDH1A1 P00352 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
CYTH2 Q99418 1/20 0.42
MCL1 Q07820 1/20 0.41
GPR35 Q9HC97 3/20 0.41
PIM1 P11309 2/20 0.41
NUAK1 O60285 1/20 0.41
IGF1R P08069 1/20 0.41
SRC P12931 1/20 0.41
KDR P35968 1/20 0.41
PLK1 P53350 1/20 0.41
PKN1 Q16512 1/20 0.41
AURKB Q96GD4 1/20 0.41
ALK Q9UM73 1/20 0.41
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL487041 0.89 ALDH1A1 (0.54) CYP3A4ACHEALDH1A1TDP1CYTH2
Formaldehyde SCHEMBL28712793 0.85 ALDH1A1 (0.50) CYP3A4ALDH1A1TDP1CYTH2MCL1
SCHEMBL231446 0.84 GPR35 (0.45) ALDH1A1TDP1GPR35TSHRALOX15
SCHEMBL31538467 0.83 GPR35 (0.50) ACHEALDH1A1TDP1MCL1GPR35
SCHEMBL31538466 0.83 GPR35 (0.50) ACHEALDH1A1TDP1MCL1GPR35
SCHEMBL11107564 0.83 GPR35 (0.50) ACHEALDH1A1TDP1MCL1GPR35
SCHEMBL6206050 0.81 CYP3A4 (0.49) CYP3A4ALDH1A1TDP1MCL1GPR35
SCHEMBL25726029 0.80 ALDH1A1 (0.41) CYP3A4ALDH1A1TDP1MCL1GPR35
SCHEMBL71098 0.79 GPR35 (0.45) ALDH1A1TDP1MCL1GPR35GRIN2D
SCHEMBL22995882 0.77 PKM (0.44) CYP3A4ALDH1A1TDP1CYTH2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2379529-B1 CGRP-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2015-06-10 EP disclosed
EP-2379529-B1 CGRP-ANTAGONISTS BOEHRINGER INGELHEIM INT (DE) 2015-06-10 EP disclosed
US-8952014-B2 Pyrimidine derivatives which are CGRP—antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-02-10 US disclosed
US-8952014-B2 Pyrimidine derivatives which are CGRP—antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-02-10 US disclosed
US-8952014-B2 Pyrimidine derivatives which are CGRP—antagonists BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2015-02-10 US disclosed
US-8853621-B2 Systems and methods extending the laserspray ionization mass spectrometry concept from atmospheric pressure to vacuum WAYNE STATE UNIVERSITY (US) 2014-10-07 US disclosed
US-20140027631-A1 Systems and Methods Extending the Laserspray Ionization Mass Spectrometry Concept from Atmospheric Pressure to Vacuum WAYNE STATE UNIVERSITY (US) 2014-01-30 US disclosed
US-20120088755-A1 Novel Compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-04-12 US disclosed
US-20120088755-A1 Novel Compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-04-12 US disclosed
US-20120088755-A1 Novel Compounds BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2012-04-12 US disclosed
EP-2379529-A1 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-10-26 EP disclosed
WO-2010070022-A1 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-24 WO disclosed
WO-2010070022-A1 NOVEL COMPOUNDS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-06-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120088755-A1 Novel Compounds SLC26A4, F12, SLCO1B3 CYP3A4 399/4885ACHE 3027/4885ALDH1A1 887/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.