SCHEMBL1286789

SCHEMBL1286789

O=C(O)C1CC12CCN(C(=O)c1ccccc1)CC2

nearest known ligand 0.58

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.53
ALDH1A1 P00352 3/20 0.52
TP53 P04637 1/20 0.52
ACHE P22303 1/20 0.51
TSHR P16473 2/20 0.51
KDM4E B2RXH2 1/20 0.51
HTT P42858 1/20 0.51
SIGMAR1 Q99720 1/20 0.50
CHRM2 P08172 1/20 0.50
CHRM3 P20309 1/20 0.50
CRBN Q96SW2 1/20 0.50
HRH3 Q9Y5N1 1/20 0.48
USP2 O75604 2/20 0.48
EPHX1 P07099 1/20 0.48
L3MBTL3 Q96JM7 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1286799 0.81 BLM (0.48) ALDH1A1ACHETSHRKDM4ECHRM2
SCHEMBL21726745 0.78 KMT2A (0.42) ALDH1A1TSHRHRH3
SCHEMBL21726748 0.78 KMT2A (0.42) ALDH1A1TSHRHRH3
SCHEMBL14812968 0.78 CYP3A4 (0.57) HPGDALDH1A1TP53TSHRUSP2
SCHEMBL1286820 0.78 HRH3 (0.59) ALDH1A1TP53TSHRHRH3USP2
SCHEMBL1709223 0.76 POLB (0.50) HPGDALDH1A1TSHR
SCHEMBL22615930 0.76 HRH3 (0.40) HRH3
SCHEMBL15655020 0.76 HRH3 (0.40) HRH3
SCHEMBL3977397 0.76 HPGD (0.58) HPGDALDH1A1TP53ACHETSHR
SCHEMBL6233435 0.76 HPGD (0.58) HPGDALDH1A1TP53ACHESIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed