SCHEMBL12879262

SCHEMBL12879262

COC(=O)c1cncc(/C=C/c2ccc(OCC3C(c4c(Cl)cccc4Cl)=NOC3C3CC3)cc2Cl)c1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
NR1H4 Q96RI1 17/20 0.41
MEN1 O00255 1/20 0.40
FABP1 P07148 1/20 0.40
THRB P10828 1/20 0.40
LIFR P42702 1/20 0.40
RECQL P46063 1/20 0.40
BLM P54132 1/20 0.40
KMT2A Q03164 1/20 0.40
HSD17B13 Q7Z5P4 1/20 0.40
RAF1 P04049 1/20 0.38
KDR P35968 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12879066 0.83 NR1H4 (0.51) NR1H4
SCHEMBL12879071 0.80 NR1H4 (0.36) NR1H4MEN1FABP1THRBLIFR
SCHEMBL12879009 0.79 NR1H4 (0.48) NR1H4
SCHEMBL12878995 0.78 NR1H4 (0.35) NR1H4MEN1FABP1THRBLIFR
SCHEMBL12879074 0.78 NR1H4 (0.33) NR1H4
SCHEMBL23474093 0.76 ACACB (0.38) NR1H4KDR
SCHEMBL12879170 0.76 NR1H4 (0.37) NR1H4MEN1FABP1THRBLIFR
SCHEMBL12188530 0.76 NR1H4 (0.69) NR1H4MEN1FABP1THRBLIFR
SCHEMBL19230732 0.75 NR1H4 (0.34) NR1H4MEN1KMT2A
SCHEMBL19620248 0.75 NR1H4 (0.51) NR1H4HSD17B13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011020615-A1 NOVEL FXR (NR1H4 ) BINDING AND ACTIVITY MODULATING COMPOUNDS PHENEX PHARMACEUTICALS AG (DE) 2011-02-24 WO disclosed