SCHEMBL1287928

SCHEMBL1287928

CCc1c(-c2ccc(F)cc2)n(COCc2ccccc2)c(=O)[nH]c1=O

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
CYP2C9 P11712 1/20 0.46
CYP2C19 P33261 1/20 0.46
RXFP1 Q9HBX9 1/20 0.41
TK1 P04183 1/20 0.39
SLC34A1 Q06495 1/20 0.38
UPP1 Q16831 1/20 0.38
SIRT2 Q8IXJ6 1/20 0.38
SIRT1 Q96EB6 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
DRD1 P21728 2/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
HPGD P15428 1/20 0.36
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2B Q13224 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1687635 0.95 ALDH1A1 (0.46) ALDH1A1CYP2C9CYP2C19RXFP1SIRT2
SCHEMBL1287915 0.82 ALDH1A1 (0.39) ALDH1A1CYP2C9CYP2C19SLC34A1L3MBTL1
SCHEMBL9597854 0.76 ALDH1A1 (0.53) ALDH1A1CYP2C9CYP2C19TK1UPP1
SCHEMBL9016369 0.76 ALDH1A1 (0.56) ALDH1A1CYP2C9CYP2C19TK1UPP1
SCHEMBL1687638 0.75 ADORA2A (0.36) ALDH1A1SLC34A1L3MBTL1HPGD
SCHEMBL1288013 0.73 UPP1 (0.59) ALDH1A1TK1UPP1HPGD
SCHEMBL8067219 0.73 ALDH1A1 (0.55) ALDH1A1CYP2C9CYP2C19TK1UPP1
SCHEMBL1287950 0.72 KMT2A (0.36) ALDH1A1CYP2C9CYP2C19L3MBTL1SMN1; SMN2
SCHEMBL10069632 0.72 ALDH1A1 (0.43) ALDH1A1SMN1; SMN2
SCHEMBL7758840 0.72 ALDH1A1 (0.51) ALDH1A1CYP2C9CYP2C19TK1UPP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047993-A2 N-HYDROXYPYRIMIDINE-2,4-DIONES AS INHIBITORS OF HIV AND HCV REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-04-12 WO disclosed
WO-2012047993-A2 N-HYDROXYPYRIMIDINE-2,4-DIONES AS INHIBITORS OF HIV AND HCV REGENTS OF THE UNIVERSITY OF MINNESOTA (US) 2012-04-12 WO disclosed