SCHEMBL12892181

SCHEMBL12892181

O=C(O)c1ccc(C2=NNNN2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44
MAP2K4 P45985 3/20 0.42
BCL2L1 Q07817 1/20 0.42
BAD Q92934 1/20 0.42
KDM4E B2RXH2 2/20 0.42
ALDH1A1 P00352 1/20 0.42
TTR P02766 1/20 0.42
SRD5A2 P31213 2/20 0.40
RXRA P19793 3/20 0.40
RXRB P28702 3/20 0.40
RAB9A P51151 2/20 0.40
RXRG P48443 1/20 0.40
MKNK1 Q9BUB5 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
NPC1 O15118 1/20 0.40
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
TOP1 P11387 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28933863 0.76 TSHR (0.52) TP53TSHRMAP2K4BCL2L1BAD
SCHEMBL19403602 0.72 ALDH1A1 (0.42) TP53KDM4EALDH1A1RAB9ANPC1
SCHEMBL14018385 0.70 TSHR (0.80) TP53TSHRBCL2L1BADALDH1A1
SCHEMBL69873 0.70 TSHR (0.80) TP53TSHRBCL2L1BADALDH1A1
SCHEMBL2637326 0.70 TSHR (0.80) TP53TSHRBCL2L1BADALDH1A1
Terephthalic Acid SCHEMBL9577834 0.70 TSHR (0.80) TP53TSHRBCL2L1BADALDH1A1
Terephthalic Acid SCHEMBL1006723 0.69 TSHR (0.92) TP53TSHRBCL2L1BADALDH1A1
Terephthalic Acid SCHEMBL9484769 0.69 TSHR (0.92) TP53TSHRBCL2L1BADALDH1A1
SCHEMBL12987957 0.67 TSHR (0.75) TP53TSHRBCL2L1BADALDH1A1
Water SCHEMBL22788424 0.67 TSHR (0.75) TP53TSHRBCL2L1BADALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7879893-B2 Zinc binding ligand; sustained release of insulin NOVO NORDISK A/S (DK) 2011-02-01 US disclosed
US-7879893-B2 Zinc binding ligand; sustained release of insulin NOVO NORDISK A/S (DK) 2011-02-01 US disclosed