SCHEMBL128943

SCHEMBL128943

COc1c(CC[N+](=O)[O-])ccc(Br)c1CO

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.38
NPC1 O15118 1/20 0.38
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
MAPT P10636 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 2/20 0.32
CYP2C19 P33261 2/20 0.32
CYP2D6 P10635 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL129011 0.84 ALDH1A1 (0.39) ALDH1A1NPC1CA2CA4MAPT
SCHEMBL16510682 0.79 SLC2A1 (0.36) ALDH1A1NPC1MAPTLMNAPOLB
SCHEMBL13077116 0.78 ALDH1A1 (0.37) ALDH1A1NPC1MAPTLMNAPOLB
SCHEMBL128806 0.78 TAAR1 (0.42) CA2CA4CYP1A2
SCHEMBL10773713 0.73 AOC3 (0.51) ALDH1A1NPC1POLBCYP2C19CYP1A2
SCHEMBL127767 0.71 PRMT1 (0.51) ALDH1A1NPC1CA2CA4MAPT
SCHEMBL22953956 0.69 CA2 (0.52) ALDH1A1CA2CA4MAPTLMNA
SCHEMBL21198523 0.68 PYCR1 (0.47) ALDH1A1NPC1MAPTLMNA
SCHEMBL30823720 0.68 PYCR1 (0.47) ALDH1A1NPC1MAPTLMNA
SCHEMBL3205488 0.65 ALDH1A1 (0.41) ALDH1A1NPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9227966-B2 Antimicrobial agents RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2016-01-05 US disclosed
US-8933096-B2 Antimicrobial agents Rugers, The State University of New Jersey (US) 2015-01-13 US disclosed
US-20140315939-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2014-10-23 US disclosed
US-20130116278-A1 ANTIMICROBIAL AGENTS RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY 2013-05-09 US disclosed
US-20120059026-A1 ANTIMICROBIAL AGENTS UNIVERSITY OF MEDICINE AND DENTISTRY OF NEW JERSEY (US) 2012-03-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130116278-A1 ANTIMICROBIAL AGENTS MRPL21, ARG1, RPP30 ALDH1A1 3341/4885NPC1 1513/4885CA2 3868/4885
US-20120059026-A1 ANTIMICROBIAL AGENTS ZYX, Q6ZSR9, ZC3HAV1L ALDH1A1 2930/4885NPC1 866/4885CA2 1379/4885
US-20140315939-A1 ANTIMICROBIAL AGENTS ZYX, Q6ZSR9, ZC3HAV1L ALDH1A1 3376/4885NPC1 799/4885CA2 1626/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.