SCHEMBL1289874

SCHEMBL1289874

Cc1ccc(C)c(-c2ncco2)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.42
HPGD P15428 2/20 0.42
KDM4E B2RXH2 2/20 0.42
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
CASP3 P42574 1/20 0.42
RAB9A P51151 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
SENP8 Q96LD8 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SENP7 Q9BQF6 1/20 0.42
SENP6 Q9GZR1 1/20 0.42
BRD4 O60885 1/20 0.40
TUBB4A P04350 2/20 0.38
TUBB P07437 2/20 0.38
TUBA3C P0DPH7 2/20 0.38
TUBA1B P68363 2/20 0.38
TUBA4A P68366 2/20 0.38
TUBB4B P68371 2/20 0.38
TUBB3 Q13509 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11017014 0.85 NPC1 (0.46) ALDH1A1HPGDKDM4EGAAMAPT
SCHEMBL4408061 0.82 KDM4E (0.43) ALDH1A1HPGDKDM4EGAAMAPT
SCHEMBL20144907 0.82 ADRA1A (0.47) BRD4TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL3725066 0.82 BRD4 (0.38) HPGDMAPTRAB9ASMN1; SMN2BRD4
SCHEMBL17102182 0.82 BRD4 (0.38) RAB9ASMN1; SMN2BRD4TUBB4ATUBB
SCHEMBL16521356 0.80 TRPA1 (0.42) HPGDGAARAB9ASMN1; SMN2BRD4
SCHEMBL8232687 0.80 IL2 (0.45) SMN1; SMN2BRD4TUBB4ATUBBTUBA3C
SCHEMBL14108017 0.80 HCRTR1 (0.46) ALDH1A1HPGDKDM4EMAPTSMN1; SMN2
SCHEMBL14951108 0.80 TUBB4A (0.47) ALDH1A1KDM4EGAASMN1; SMN2TUBB4A
SCHEMBL22187760 0.79 CTSA (0.44) BRD4TUBB4ATUBBTUBA3CTUBA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 32 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209747-A1 NEW CLASS OF ORGANIC PHOSPHORS BASED ON DERIVATIVES OF BENZIMIDAZOXANTHENOISOQUINOLINONE FOR LED LIGHTING Philips Lighting Holding B.V. (NL) 2017-08-30 EP disclosed
EP-2663551-A1 NEW FLUORESCENT COMPOUNDS BASF SE (DE) 2013-11-20 EP disclosed
EP-2625171-A1 PHENANTHRO[9,10-B]FURANS FOR ELECTRONIC APPLICATIONS BASF SE (DE) 2013-08-14 EP disclosed
EP-2582769-A1 ORGANIC ELECTRONIC DEVICES COMPRISING A LAYER OF A DIBENZOFURANE COMPOUND AND A 8-HYDROXYQUINOLINOLATO EARTH ALKALINE METAL, OR ALKALI METAL COMPLEX BASF SE (DE) 2013-04-24 EP disclosed
EP-2582768-A1 ORGANIC ELECTRONIC DEVICES COMPRISING A LAYER OF A PYRIDINE COMPOUND AND A 8-HYDROXYQUINOLINOLATO EARTH ALKALINE METAL, OR ALKALI METAL COMPLEX BASF SE (DE) 2013-04-24 EP disclosed
EP-2582770-A1 ORGANIC ELECTRONIC DEVICES COMPRISING THE LAYER CONTAINING AT LEAST ONE METAL ORGANIC COMPOUND AND AT LEAST ONE METAL OXIDE BASF SE (DE) 2013-04-24 EP disclosed
WO-2012095803-A1 NEW FLUORESCENT COMPOUNDS BASF SE (DE) 2012-07-19 WO disclosed
WO-2012045710-A1 PHENANTHRO[9,10-B]FURANS FOR ELECTRONIC APPLICATIONS BASF SE (DE) 2012-04-12 WO disclosed
WO-2011157790-A1 ORGANIC ELECTRONIC DEVICES COMPRISING A LAYER OF A DIBENZOFURANE COMPOUND AND A 8-HYDROXYQUINOLINOLATO EARTH ALKALINE METAL, OR ALKALI METAL COMPLEX BASF SE (DE) 2011-12-22 WO disclosed
WO-2011158204-A1 ORGANIC ELECTRONIC DEVICES COMPRISING THE LAYER CONTAINING AT LEAST ONE METAL ORGANIC COMPOUND AND AT LEAST ONE METAL OXIDE BASF SE (DE) 2011-12-22 WO disclosed
EP-1981929-A1 NOVEL POLYMERS Ciba Holding Inc. (CH) 2008-10-22 EP disclosed
WO-2008119666-A1 HETEROCYCLIC BRIDGED BIPHENYLS BASF SE (CH) 2008-10-09 WO disclosed
WO-2008031743-A1 HETEROCYCLIC BRIDGED BIPHENYLS AND THEIR USE IN OLEDS CIBA HOLDING INC. (CH) 2008-03-20 WO disclosed
WO-2008012250-A1 NOVEL POLYMERS CIBA HOLDING INC. (CH) 2008-01-31 WO disclosed
WO-2008006743-A1 NOVEL ELECTROLUMINESCENT POLYMERS FOR ELECTRONIC APPLICATIONS CIBA HOLDING INC (CH) 2008-01-17 WO disclosed
EP-1858976-A1 NOVEL POLYMERS Ciba Specialty Chemicals Holding Inc. (CH) 2007-11-28 EP disclosed
WO-2007090773-A1 NOVEL POLYMERS CIBA HOLDING INC. (CH) 2007-08-16 WO disclosed
WO-2006097419-A1 NOVEL POLYMERS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2006-09-21 WO disclosed
EP-1682605-A1 NOVEL DIKETOPYRROLOPYRROLE POLYMERS Ciba SC Holding AG (CH) 2006-07-26 EP disclosed
WO-2005049695-A1 NOVEL DIKETOPYRROLOPYRROLE POLYMERS CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2005-06-02 WO disclosed