SCHEMBL20144907

SCHEMBL20144907

Cc1ccc(F)cc1-c1ncco1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 2/20 0.47
HCRTR1 O43613 3/20 0.44
HCRTR2 O43614 2/20 0.44
NISCH Q9Y2I1 1/20 0.44
ADRA2A P08913 1/20 0.43
ADRA1D P25100 1/20 0.43
ADRA1B P35368 1/20 0.43
ABL1 P00519 3/20 0.39
IL2 P60568 1/20 0.39
TUBB4A P04350 1/20 0.38
TUBB P07437 1/20 0.38
TUBA3C P0DPH7 1/20 0.38
TUBA1B P68363 1/20 0.38
TUBA4A P68366 1/20 0.38
TUBB4B P68371 1/20 0.38
TUBB3 Q13509 1/20 0.38
TUBB2A Q13885 1/20 0.38
TUBB8 Q3ZCM7 1/20 0.38
TUBA3E Q6PEY2 1/20 0.38
TUBA1A Q71U36 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1289874 0.82 ALDH1A1 (0.42) IL2TUBB4ATUBBTUBA3CTUBA1B
SCHEMBL4408061 0.79 KDM4E (0.43) IL2BRD4PIK3CDPIK3CGHPGDS
SCHEMBL17102182 0.79 BRD4 (0.38) HCRTR1HCRTR2IL2TUBB4ATUBB
SCHEMBL31039212 0.79 ADRA1A (0.47) ADRA1AHCRTR1HCRTR2ADRA2AADRA1D
SCHEMBL7834048 0.79 ADRA1A (0.48) ADRA1AHCRTR1HCRTR2ADRA2AADRA1D
SCHEMBL14108017 0.77 HCRTR1 (0.46) ADRA1AHCRTR1HCRTR2NISCHADRA2A
SCHEMBL16149099 0.76 HCRTR1 (0.52) ADRA1AHCRTR1HCRTR2ADRA2AADRA1D
SCHEMBL3031254 0.74 RAB9A (0.53) ADRA1AADRA2AADRA1DADRA1BBRD4
SCHEMBL4265596 0.73 ALDH1A1 (0.49) PDE2A
SCHEMBL22187760 0.72 CTSA (0.44) ADRA1AHCRTR1HCRTR2ADRA2AADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2970207-B1 SUBSTITUTED PIPERIDINE COMPOUNDS AND THEIR USE AS OREXIN RECEPTOR MODULATORS JANSSEN PHARMACEUTICA NV (BE) 2018-05-16 EP disclosed