SCHEMBL12901062

SCHEMBL12901062

Cc1cc(Nc2cccnc2)c(C(F)(F)F)cn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.50
IL1B P01584 1/20 0.41
NLRP3 Q96P20 1/20 0.41
CTSC P53634 1/20 0.41
TSHR P16473 2/20 0.41
NOTUM Q6P988 1/20 0.40
GRM5 P41594 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CCNK O75909 1/20 0.38
CCNA2 P20248 1/20 0.38
CDK2 P24941 1/20 0.38
CCND3 P30281 1/20 0.38
CDK9 P50750 1/20 0.38
CDK6 Q00534 1/20 0.38
BRAF P15056 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1231857 0.83 KIF11 (0.50) KIF11CTSCTSHRNOTUML3MBTL1
SCHEMBL29801195 0.76 KIF11 (0.54) KIF11TSHRNOTUML3MBTL1ALDH1A1
SCHEMBL12901052 0.76 MEN1 (0.49) CTSCTSHRCCNKCCNA2CDK2
SCHEMBL12901776 0.74 CYP1A2 (0.41) TSHRALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL12900858 0.71 MAPK10 (0.48) MAPK8MAPK10
SCHEMBL12902136 0.71 MAPK3 (0.51) MAPK10
SCHEMBL12901097 0.70 MAPK10 (0.47) MAPK8MAPK10
SCHEMBL12901056 0.69 MAPK10 (0.58) MAPK8MAPK10
SCHEMBL12900857 0.69 NTRK1 (0.43) ALDH1A1CYP1A2CYP3A4CYP2C19MAPK8
SCHEMBL12900855 0.69 MAPK10 (0.45) TSHRALDH1A1MAPK8MAPK10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110046121-A1 INHIBITORS OF FOCAL ADHESION KINASE THE SCRIPPS RESEARCH INSTITUTE (US) 2011-02-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110046121-A1 INHIBITORS OF FOCAL ADHESION KINASE PTK2, CABLES1, TNK2 KIF11 1040/4885IL1B 4318/4885NLRP3 4619/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.