SCHEMBL12945621

SCHEMBL12945621

C=CCc1ccccc1NS(=O)(=O)c1cccc(OC)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 2/20 0.61
NFE2L2 Q16236 2/20 0.61
PGR P06401 3/20 0.55
GLO1 Q04760 1/20 0.53
SLC40A1 Q9NP59 1/20 0.53
PTGES2 Q9H7Z7 1/20 0.52
FFAR4 Q5NUL3 2/20 0.51
PGAM1 P18669 1/20 0.49
SLC16A3 O15427 1/20 0.48
TRIM24 O15164 1/20 0.48
BRD1 O95696 1/20 0.48
BRPF1 P55201 1/20 0.48
GAA P10253 1/20 0.47
HDAC3 O15379 1/20 0.47
HDAC4 P56524 1/20 0.47
HDAC1 Q13547 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12945230 0.86 KEAP1 (0.60) KEAP1NFE2L2PGRFFAR4GAA
SCHEMBL28655832 0.81 KEAP1 (0.50) KEAP1
SCHEMBL3555853 0.79 KEAP1 (0.56) KEAP1NFE2L2PGRGLO1SLC40A1
SCHEMBL3560551 0.78 KEAP1 (0.54) KEAP1NFE2L2PGRGLO1SLC40A1
SCHEMBL3557703 0.77 KEAP1 (0.53) KEAP1NFE2L2PGRGLO1SLC40A1
SCHEMBL8419064 0.77 LMNA (0.59) KEAP1NFE2L2GAA
SCHEMBL30026801 0.77 LMNA (0.59) KEAP1NFE2L2GAA
SCHEMBL17388819 0.77 PTGDR2 (0.57) KEAP1NFE2L2PGRGLO1SLC40A1
SCHEMBL28389707 0.77 FFAR4 (0.60) KEAP1NFE2L2FFAR4TRIM24BRPF1
SCHEMBL12945620 0.76 ALDH1A1 (0.45) KEAP1NFE2L2PGRFFAR4GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009059-A2 METHOD OF TREATING OR PREVENTING CANCER THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-01-20 WO disclosed