SCHEMBL12945620

SCHEMBL12945620

C=CCc1ccccc1NS(=O)(=O)Nc1ccc(OC)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.45
LMNA P02545 2/20 0.45
FFAR4 Q5NUL3 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
ALOX12 P18054 2/20 0.43
PGR P06401 2/20 0.43
TP53 P04637 1/20 0.43
CYP3A4 P08684 1/20 0.43
ALOX15 P16050 1/20 0.43
TSHR P16473 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
KEAP1 Q14145 2/20 0.41
TUBB4A P04350 1/20 0.41
TUBB P07437 1/20 0.41
TUBA3C P0DPH7 1/20 0.41
TUBA1B P68363 1/20 0.41
TUBA4A P68366 1/20 0.41
TUBB4B P68371 1/20 0.41
TUBB3 Q13509 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12945429 0.84 SLC40A1 (0.46) ALDH1A1LMNACA1CA2ALOX12
SCHEMBL12945230 0.84 KEAP1 (0.60) ALDH1A1LMNAFFAR4PGRTP53
SCHEMBL12945432 0.82 CA1 (0.40) ALDH1A1CA1CA2PGRGAA
SCHEMBL12945621 0.76 KEAP1 (0.61) FFAR4PGRKEAP1GAANFE2L2
SCHEMBL8420054 0.75 KEAP1 (0.46) ALDH1A1PGRKEAP1GAAKMT2A
SCHEMBL31011735 0.73 MAPT (0.49) ALDH1A1ALOX12TP53CYP3A4ALOX15
SCHEMBL5130307 0.72 GABRA1 (0.41) ALDH1A1LMNAALOX12TSHRSMN1; SMN2
SCHEMBL12945430 0.71 CA2 (0.53) ALDH1A1LMNACA1CA2SMN1; SMN2
SCHEMBL28655832 0.70 KEAP1 (0.50) ALDH1A1TSHRSMN1; SMN2KEAP1KMT2A
SCHEMBL9179590 0.69 TGM2 (0.59) ALDH1A1LMNACA1CA2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011009059-A2 METHOD OF TREATING OR PREVENTING CANCER THE UNITED STATES OF AMERICA, AS REPRESENTED BY THE SECRETARY, DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 2011-01-20 WO disclosed