SCHEMBL12951709

SCHEMBL12951709

NC(=O)CCCCCn1c2c(c3ccccc31)CCNC2

nearest known ligand 0.55

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 7/20 0.55
HDAC1 Q13547 6/20 0.55
BRD4 O60885 1/20 0.48
KDM4E B2RXH2 2/20 0.47
ALDH1A1 P00352 1/20 0.47
HTR6 P50406 2/20 0.46
MAOA P21397 4/20 0.45
MAOB P27338 4/20 0.45
FABP4 P15090 1/20 0.45
FABP5 Q01469 1/20 0.45
HTR2A P28223 1/20 0.44
HTR2C P28335 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12951710 0.85 HDAC6 (0.49) HDAC6HDAC1BRD4KDM4EMAOA
SCHEMBL9615110 0.82 NPC1 (0.54) HDAC6HDAC1KDM4EALDH1A1HTR6
Hydrochloric Acid SCHEMBL9615105 0.81 KDM4E (0.53) HDAC6HDAC1KDM4EALDH1A1HTR6
SCHEMBL928866 0.80 HTR6 (0.52) HDAC6HDAC1KDM4EALDH1A1HTR6
SCHEMBL46293 0.78 HDAC1 (0.52) HDAC6HDAC1KDM4EHTR6HTR2A
SCHEMBL4300297 0.77 HDAC1 (0.53) HDAC6HDAC1KDM4EALDH1A1HTR6
Trifluoroacetic Acid SCHEMBL6425706 0.77 HDAC6 (0.52) HDAC6HDAC1KDM4EALDH1A1HTR6
Hydrochloric Acid SCHEMBL14892472 0.77 HDAC1 (0.51) HDAC6HDAC1KDM4EHTR6HTR2A
SCHEMBL20961100 0.77 KDM4E (0.77) HDAC6HDAC1KDM4EMAOAMAOB
SCHEMBL20961263 0.75 KDM4E (0.80) HDAC6HDAC1KDM4EMAOAMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011011186-A2 HDAC INHIBITORS AND THERAPEUTIC METHODS USING THE SAME THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ILLINOIS (US) 2011-01-27 WO disclosed