SCHEMBL12986930

SCHEMBL12986930

CC(=O)Oc1ccccc1C(=O)OCc1ncccc1C(=O)NCCO[N+](=O)[O-]

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 4/20 0.58
HSD17B10 Q99714 4/20 0.44
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
CYP2C9 P11712 2/20 0.44
ALOX15 P16050 1/20 0.44
CYP2C19 P33261 1/20 0.44
LMNA P02545 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
MAPK1 P28482 2/20 0.40
NPC1 O15118 1/20 0.40
MLNR O43193 1/20 0.40
NR1I2 O75469 1/20 0.40
ABCB11 O95342 1/20 0.40
TP53 P04637 1/20 0.40
ADRB2 P07550 1/20 0.40
CHRM2 P08172 1/20 0.40
ADRB1 P08588 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9545778 0.83 PTGS2 (0.62) PTGS2HSD17B10MEN1KMT2ACYP2C9
SCHEMBL13588988 0.82 PTGS2 (0.58) PTGS2HSD17B10MEN1KMT2ACYP2C9
SCHEMBL12987782 0.81 MEN1 (0.49) HSD17B10MEN1KMT2ACYP2C9ALOX15
SCHEMBL12986933 0.79 KMT2A (0.47) HSD17B10MEN1KMT2ACYP2C9ALOX15
SCHEMBL12987053 0.79 KMT2A (0.47) PTGS2HSD17B10MEN1KMT2ACYP2C9
SCHEMBL12986889 0.79 KMT2A (0.47) HSD17B10MEN1KMT2ACYP2C9ALOX15
SCHEMBL12986566 0.79 MEN1 (0.47) HSD17B10MEN1KMT2ACYP2C9ALOX15
SCHEMBL4553089 0.77 PTGS2 (0.67) PTGS2HSD17B10MEN1KMT2ALMNA
SCHEMBL15639697 0.76 SYK (0.45) PTGS2HSD17B10CYP2C9LMNAALDH1A1
SCHEMBL15889887 0.76 PTGS2 (0.85) PTGS2HSD17B10MEN1KMT2ACYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2693876-A1 SUBSTITUTED METHYLFORMYL REAGENTS AND METHOD OF USING SAME TO MODIFY PHYSICOCHEMICAL AND/OR PHARMACOKINETIC PROPERTIES OF COMPOUNDS Sphaera Pharma Pte. Ltd (SG) 2014-02-12 EP claimed
WO-2012137225-A1 SUBSTITUTED METHYLFORMYL REAGENTS AND METHOD OF USING SAME TO MODIFY PHYSICOCHEMICAL AND/OR PHARMACOKINETIC PROPERTIES OF COMPOUNDS SPHAERA PHARMA PVT. LTD (IN) 2012-10-11 WO claimed