SCHEMBL13005448

SCHEMBL13005448

CCN1CCC[C@@H]1CNC(=O)c1cccc(-c2cccc(CC(C)C)c2)c1

nearest known ligand 0.56

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.53
ROCK2 O75116 2/20 0.53
ROCK1 Q13464 2/20 0.53
DRD2 P14416 4/20 0.53
ABCG2 Q9UNQ0 1/20 0.52
MCHR2 Q969V1 1/20 0.50
MCHR1 Q99705 1/20 0.50
KMT2A Q03164 1/20 0.49
HSD17B10 Q99714 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13005433 1.00 HTR1A (0.53) HTR1AROCK2ROCK1DRD2ABCG2
SCHEMBL13060677 0.90 DRD2 (0.60) HTR1AROCK2ROCK1DRD2ABCG2
SCHEMBL13060652 0.90 DRD2 (0.60) HTR1AROCK2ROCK1DRD2ABCG2
SCHEMBL19954197 0.83 ROCK2 (0.59) HTR1AROCK2ROCK1DRD2ABCG2
SCHEMBL13006797 0.82 ABCG2 (0.57) ROCK2ROCK1DRD2ABCG2KMT2A
SCHEMBL13005425 0.82 ABCG2 (0.57) ROCK2ROCK1DRD2ABCG2KMT2A
SCHEMBL13005479 0.81 ABCG2 (0.49) ROCK2ROCK1DRD2ABCG2MCHR2
SCHEMBL17790224 0.81 ROCK2 (0.61) HTR1AROCK2ROCK1DRD2ABCG2
SCHEMBL18901194 0.80 ROCK2 (0.60) HTR1AROCK2ROCK1DRD2ABCG2
SCHEMBL13005478 0.79 ABCG2 (0.47) ROCK2ROCK1DRD2ABCG2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed