SCHEMBL13005476

SCHEMBL13005476

CC(C)Cc1cccc(-c2ccc(C(=O)N(C)C)cc2)c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD17B2 P37059 5/20 0.51
HSD17B1 P14061 3/20 0.51
BCL2 P10415 1/20 0.49
AOC3 Q16853 6/20 0.48
ERN1 O75460 1/20 0.46
PTGES O14684 1/20 0.45
PTGS2 P35354 1/20 0.45
ALDH1A1 P00352 1/20 0.45
MAPT P10636 1/20 0.45
CTSL P07711 1/20 0.44
CTSB P07858 1/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
HDAC8 Q9BY41 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13005458 0.86 HPGD (0.61) HSD17B2HSD17B1BCL2AOC3PTGES
SCHEMBL23514718 0.86 ERN1 (0.52) HSD17B2HSD17B1ERN1
SCHEMBL13060851 0.84 BCL2 (0.69) HSD17B2HSD17B1BCL2AOC3ERN1
SCHEMBL10160068 0.83 KMT2A (0.49) HSD17B2HSD17B1ERN1
SCHEMBL8180284 0.80 ACACB (0.56) PTGS2ALDH1A1
SCHEMBL13005470 0.78 ERN1 (0.47) ERN1ALDH1A1
SCHEMBL13680801 0.78 ERN1 (0.50) HSD17B2HSD17B1BCL2AOC3ERN1
SCHEMBL8636391 0.78 MEN1 (0.46) BCL2PTGS2MAPTCTSSCTSK
SCHEMBL28161128 0.78 CTSS (0.48) PTGS2CTSSCTSK
SCHEMBL1513819 0.77 MMP3 (0.56) HSD17B2HSD17B1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed