SCHEMBL13005491

SCHEMBL13005491

CC(C)Cc1cccc(C(=O)N[C@H](Cc2ccccc2)CN(C)C)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTRB1 P17538 1/20 0.51
HDAC4 P56524 4/20 0.50
HDAC6 Q9UBN7 4/20 0.50
MME P08473 1/20 0.49
MMEL1 Q495T6 1/20 0.49
PIN1 Q13526 2/20 0.46
HDAC1 Q13547 1/20 0.46
CTSL P07711 1/20 0.45
ALDH1A1 P00352 1/20 0.45
SLC7A5 Q01650 1/20 0.44
ECE1 P42892 1/20 0.44
FOLH1 Q04609 1/20 0.43
CTSD P07339 1/20 0.43
BACE1 P56817 1/20 0.43
BACE2 Q9Y5Z0 1/20 0.43
GPR139 Q6DWJ6 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
GPR132 Q9UNW8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13005665 0.93 MME (0.51) CTRB1HDAC4HDAC6MMEMMEL1
SCHEMBL13005584 0.90 KMT2A (0.51) CTRB1HDAC4HDAC6ALDH1A1
SCHEMBL13061025 0.89 CTRB1 (0.52) CTRB1HDAC4HDAC6MMEMMEL1
SCHEMBL23116558 0.87 CTRB1 (0.66) CTRB1HDAC4HDAC6PIN1HDAC1
SCHEMBL10952300 0.87 CTRB1 (0.66) CTRB1HDAC4HDAC6PIN1HDAC1
SCHEMBL13005579 0.83 KMT2A (0.47) CTRB1MMEMMEL1CTSL
SCHEMBL13060697 0.82 MME (0.52) CTRB1HDAC4HDAC6MMEMMEL1
SCHEMBL13005434 0.82 HDAC4 (0.45) HDAC4MMEMMEL1CTSLALDH1A1
SCHEMBL13005436 0.82 HDAC4 (0.45) HDAC4MMEMMEL1CTSLALDH1A1
SCHEMBL13005496 0.80 MME (0.43) CTRB1HDAC4HDAC6MMEMMEL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed