SCHEMBL13005492

SCHEMBL13005492

CC(C)Cc1cccc(CN([C@@H](Cc2ccccc2)CN(C)C)S(C)(=O)=O)c1

nearest known ligand 0.50

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
CETP P11597 1/20 0.38
ALOX5 P09917 1/20 0.36
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
SLC6A2 P23975 1/20 0.35
HTR2A P28223 1/20 0.35
SLC6A4 P31645 1/20 0.35
ADRA1A P35348 1/20 0.35
OPRK1 P41145 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KCNH2 Q12809 1/20 0.35
HPGD P15428 1/20 0.35
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13061016 0.89 TSHR (0.40) TSHRADRA2BADRA2CSLC6A2HTR2A
SCHEMBL13005487 0.82 CETP (0.40) TSHRCETPALOX5ADRA2BADRA2C
SCHEMBL13005484 0.82 OPRK1 (0.47) CETPALOX5ADRA2BADRA2CSLC6A2
SCHEMBL13005495 0.81 OPRK1 (0.43) TSHRCETPALOX5ADRA2BADRA2C
SCHEMBL13005494 0.79 ALOX5 (0.41) CETPALOX5HPGD
SCHEMBL13005518 0.74 CETP (0.40) TSHRCETPALOX5ADRA2BADRA2C
SCHEMBL13005557 0.72 SIGMAR1 (0.41) TSHRCETPALOX5ADRA2BADRA2C
SCHEMBL13005605 0.72 SLC6A2 (0.45) TSHRCETPALOX5ADRA2BADRA2C
SCHEMBL13060671 0.72 OPRK1 (0.39) TSHRADRA2BADRA2CSLC6A2HTR2A
SCHEMBL16640979 0.72 ALDH1A1 (0.50) TSHRCETPADRA2BADRA2CSLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed