SCHEMBL13005507

SCHEMBL13005507

CC(C)Cc1cccc(CN(Cc2ccccc2Br)[C@@H](CC(C)C)CN(C)C)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.34
CETP P11597 1/20 0.34
PYCR1 P32322 1/20 0.33
TSHR P16473 2/20 0.32
GRIN2D O15399 1/20 0.32
GRIN3B O60391 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2A Q12879 1/20 0.32
GRIN2B Q13224 1/20 0.32
GRIN2C Q14957 1/20 0.32
GRIN3A Q8TCU5 1/20 0.32
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
NFKB1 P19838 1/20 0.30
CYP2C19 P33261 1/20 0.30
HSD17B10 Q99714 1/20 0.30
ANPEP P15144 1/20 0.30
MMP2 P08253 1/20 0.30
MMP3 P08254 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13061103 0.92 TSHR (0.35) TAAR1PYCR1TSHRGRIN2DGRIN3B
SCHEMBL13005518 0.87 CETP (0.40) TAAR1CETPTSHRGRIN2DGRIN3B
SCHEMBL13005522 0.86 CETP (0.36) CETPGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL13005520 0.86 LMNA (0.37) TAAR1CETPPYCR1LMNA
SCHEMBL13005500 0.86 GABRA1 (0.39) CETPGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL13005504 0.86 ALDH1A1 (0.36) TAAR1CETPGRIN2DGRIN3BGRIN1
SCHEMBL13005616 0.84 BCHE (0.40) CETPCYP2D6
SCHEMBL13005513 0.84 CETP (0.32) CETPGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL13005551 0.83 CETP (0.35) TAAR1CETPPYCR1TSHRGRIN2D
SCHEMBL13005523 0.83 TAAR1 (0.36) TAAR1CETPPYCR1TSHRGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed