SCHEMBL13005702

SCHEMBL13005702

CC(C)Cc1cccc(CN(CCN(C)C)Cc2cccc(Br)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.53
CALM1 P0DP23 1/20 0.46
CAMKK2 Q96RR4 1/20 0.46
PYCR1 P32322 1/20 0.43
SIGMAR1 Q99720 3/20 0.42
PTGES O14684 1/20 0.40
ACKR3 P25106 1/20 0.40
RIPK1 Q13546 1/20 0.39
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
BCHE P06276 1/20 0.35
TSHR P16473 1/20 0.35
RECQL P46063 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13005681 0.90 CALM1 (0.48) TAAR1CALM1CAMKK2PYCR1PTGES
SCHEMBL13005440 0.87 CALM1 (0.59) TAAR1CALM1CAMKK2MEN1KMT2A
SCHEMBL13005625 0.85 BCHE (0.47) TAAR1CALM1CAMKK2MEN1KMT2A
SCHEMBL13061011 0.84 TAAR1 (0.57) TAAR1CALM1CAMKK2PYCR1SIGMAR1
SCHEMBL14181862 0.84 CALM1 (0.62) TAAR1CALM1CAMKK2PYCR1SIGMAR1
SCHEMBL13005684 0.83 TAAR1 (0.53) TAAR1CALM1CAMKK2RIPK1MEN1
SCHEMBL13005692 0.83 TSHR (0.54) TAAR1CALM1CAMKK2PYCR1RIPK1
SCHEMBL13005720 0.83 OPRK1 (0.49) CALM1CAMKK2MEN1KMT2A
SCHEMBL13005422 0.83 CALM1 (0.48) TAAR1CALM1CAMKK2MEN1KMT2A
SCHEMBL14027648 0.82 TAAR1 (0.58) TAAR1CALM1CAMKK2PYCR1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed