SCHEMBL13014116

SCHEMBL13014116

CN1CCN(CC(=O)O)CCN(CC(=O)O)CCN(CC(CCCc2ccc(N)cc2)N(CC(=O)O)CC(=O)O)CC1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 1/20 0.41
LMNA P02545 1/20 0.40
SIGMAR1 Q99720 3/20 0.39
OPRK1 P41145 1/20 0.35
MC4R P32245 3/20 0.34
KMT2A Q03164 1/20 0.33
PPARG P37231 1/20 0.33
PPARA Q07869 1/20 0.33
POLB P06746 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
GAA P10253 1/20 0.33
ALB P02768 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM4 P08173 1/20 0.32
NOS3 P29474 1/20 0.32
NOS1 P29475 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18079519 0.95 S1PR1 (0.42) S1PR1SIGMAR1OPRK1ALBCHRM2
SCHEMBL3779770 0.95 S1PR1 (0.42) S1PR1SIGMAR1OPRK1ALBCHRM2
SCHEMBL18022816 0.91 S1PR1 (0.46) S1PR1SIGMAR1OPRK1ALB
SCHEMBL27404859 0.89 SIGMAR1 (0.39) S1PR1SIGMAR1OPRK1CHRM2CHRM4
SCHEMBL13014130 0.86 KCNJ1 (0.45) SIGMAR1OPRK1KMT2A
SCHEMBL13014054 0.86 KCNJ1 (0.45) SIGMAR1OPRK1KMT2A
SCHEMBL24618857 0.86 SIGMAR1 (0.50) SIGMAR1MC4RKMT2APOLBGAA
SCHEMBL24240930 0.85 S1PR1 (0.42) S1PR1LMNASIGMAR1KMT2APOLB
SCHEMBL26241146 0.85 OPRD1 (0.41) S1PR1SIGMAR1KMT2A
SCHEMBL22821437 0.83 S1PR1 (0.42) S1PR1KMT2APOLBGAAALB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9115094-B2 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using THE UNITED STATES OF AMERICA, NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS) (US) 2015-08-25 US disclosed
US-20100322855-A1 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using ILLINOIS INSTITUTE OF TECHNOLOGY (US) 2010-12-23 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100322855-A1 Bimodal ligands with macrocyclic and acyclic binding moieties, complexes and compositions thereof, and methods of using UACA, CLTC, PKD1 S1PR1 2492/4885LMNA 559/4885SIGMAR1 870/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.