SCHEMBL13014248

SCHEMBL13014248

CCOC(=O)C1=C(C)Nc2c(c(Nc3ccc(Cl)cc3)nc(=O)n2-c2ccccc2)C1c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABCC1 P33527 1/20 0.48
ADORA3 P0DMS8 1/20 0.46
ACHE P22303 2/20 0.44
CACNA1D Q01668 1/20 0.43
KDM4E B2RXH2 3/20 0.43
ALDH1A1 P00352 3/20 0.43
NPEPPS P55786 1/20 0.43
KDM4A O75164 1/20 0.43
USP2 O75604 1/20 0.43
MPI P34949 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
HPGD P15428 2/20 0.42
CASP3 P42574 1/20 0.42
MAPT P10636 2/20 0.42
HTT P42858 1/20 0.41
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
DHODH Q02127 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13014429 0.95 ADORA3 (0.51) ADORA3ACHECACNA1DKDM4EALDH1A1
SCHEMBL3433331 0.93 CASP3 (0.49) ADORA3ACHEKDM4EALDH1A1NPEPPS
SCHEMBL13013473 0.90 HPGD (0.49) ABCC1ADORA3ACHECACNA1DKDM4E
SCHEMBL13014289 0.90 ALDH1A1 (0.44) ABCC1ACHECACNA1DKDM4EALDH1A1
SCHEMBL13013458 0.90 ADORA3 (0.44) ABCC1ADORA3ACHEKDM4EALDH1A1
SCHEMBL13012935 0.89 ADORA3 (0.49) ABCC1ADORA3ACHECACNA1DKDM4E
SCHEMBL13013490 0.88 ADORA3 (0.48) ABCC1ADORA3ACHECACNA1DKDM4E
SCHEMBL13013560 0.87 ADORA3 (0.46) ADORA3ACHEKDM4EALDH1A1MAPT
SCHEMBL13014273 0.87 ADORA3 (0.47) ABCC1ADORA3ACHECACNA1DKDM4E
SCHEMBL13013037 0.87 ABCC1 (0.46) ABCC1ADORA3ACHECACNA1DKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010149786-A1 PYRIDO [2, 3-D] PYRIMIDINES AS WNT ANTAGONISTS FOR TREATMENT OF CANCER AND ARTHRITIS DEUTSCHES KREBSFORSCHUNGSZENTRUM (DE) 2010-12-29 WO disclosed