SCHEMBL13044524

SCHEMBL13044524

Cc1cc(C)cc(NNC(=O)C(c2ccc3ccccc3c2)N2CCN(C)CC2)c1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.48
ABCB1 P08183 10/20 0.47
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
LMNA P02545 1/20 0.41
SLC1A3 P43003 1/20 0.40
SLC1A2 P43004 1/20 0.40
HPGD P15428 1/20 0.40
TSHR P16473 1/20 0.40
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPT P10636 1/20 0.39
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3639856 0.88 GHSR (0.52) GHSRABCB1KMT2AMEN1LMNA
SCHEMBL13044525 0.85 GHSR (0.68) GHSRABCB1KMT2ASLC1A3SLC1A2
Formic Acid SCHEMBL3737845 0.85 GHSR (0.49) GHSRABCB1KMT2AMEN1LMNA
SCHEMBL3639221 0.82 GHSR (0.55) GHSRABCB1KMT2AMEN1ALDH1A1
SCHEMBL13044326 0.77 HPGD (0.50) ABCB1LMNASLC1A3SLC1A2HPGD
SCHEMBL3639648 0.77 CLK1 (0.46) GHSRKMT2AMEN1LMNATSHR
Hydrochloric Acid SCHEMBL3637935 0.76 LMNA (0.51) ABCB1LMNASLC1A3SLC1A2HPGD
SCHEMBL3634225 0.74 GHSR (0.67) GHSRABCB1KMT2AMEN1LMNA
SCHEMBL3638220 0.73 GHSR (0.53) GHSRABCB1KMT2AMEN1LMNA
SCHEMBL3637462 0.73 GHSR (0.46) GHSRABCB1KMT2AMEN1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20100286152-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2010-11-11 US disclosed
US-20100286152-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2010-11-11 US disclosed
WO-2008148853-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GLAXO GROUP LIMITED (GB) 2008-12-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100286152-A1 N-PHENYL HYDRAZIDES AS MODULATORS OF THE GHRELIN RECEPTOR GIPR, GHSR, GLP1R GHSR 2/4885ABCB1 2178/4885KMT2A 3646/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.