SCHEMBL13048833

SCHEMBL13048833

C=CC(=O)Nc1sc(-c2cncc(F)c2)nc1C#N

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CG P48736 2/20 0.38
DYRK1A Q13627 5/20 0.38
TBK1 Q9UHD2 1/20 0.36
GSTO1 P78417 2/20 0.34
CYP11B1 P15538 1/20 0.34
CYP11B2 P19099 1/20 0.34
TGM2 P21980 1/20 0.33
HDAC6 Q9UBN7 1/20 0.32
EGFR P00533 1/20 0.32
ITK Q08881 1/20 0.32
ABL1 P00519 2/20 0.32
BTK Q06187 1/20 0.31
PIM1 P11309 1/20 0.31
KDR P35968 1/20 0.31
TEK Q02763 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13074603 0.83 PIK3CG (0.40) PIK3CGDYRK1AGSTO1TGM2EGFR
SCHEMBL289594 0.78 ALOX15 (0.46) PIK3CGDYRK1ATBK1CYP11B1CYP11B2
SCHEMBL13048814 0.78 TBK1 (0.39) PIK3CGDYRK1ATBK1CYP11B1CYP11B2
SCHEMBL15109438 0.77 TBK1 (0.38) PIK3CGDYRK1ATBK1CYP11B1CYP11B2
SCHEMBL25405384 0.69 PIK3CG (0.44) PIK3CGDYRK1AABL1PIM1
SCHEMBL18569065 0.69 CYP11B1 (0.40) PIK3CGDYRK1ACYP11B1CYP11B2
SCHEMBL13075078 0.66 DYRK1A (0.47) PIK3CGDYRK1AABL1PIM1
SCHEMBL13047720 0.65 DYRK1A (0.43) PIK3CGDYRK1AABL1PIM1
SCHEMBL290286 0.65 TRPM8 (0.32) PIK3CGDYRK1ACYP11B1CYP11B2
SCHEMBL18569322 0.64 CYP1A2 (0.38) PIK3CGDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 19 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2614826-B1 Process for preparation of thiazole derivatives DOW AGROSCIENCES LLC (US) 2017-03-01 EP disclosed
US-9006446-B2 Pesticidal compositions DOW AGROSCIENCES LLC (US) 2015-04-14 US disclosed
US-9006446-B2 Pesticidal compositions DOW AGROSCIENCES LLC (US) 2015-04-14 US disclosed
US-20150045218-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2015-02-12 US disclosed
US-20150045218-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2015-02-12 US disclosed
US-8853246-B2 Pesticidal compositions DOW AGROSCIENCES, LLC. (US) 2014-10-07 US disclosed
US-8853246-B2 Pesticidal compositions DOW AGROSCIENCES, LLC. (US) 2014-10-07 US disclosed
EP-2614826-A1 Process for preparation of thiazole derivatives Dow AgroSciences LLC (US) 2013-07-17 EP disclosed
EP-2614825-A1 Process for the preparation of thiazole derivatives Dow AgroSciences LLC (US) 2013-07-17 EP disclosed
EP-2604267-A1 Process for the preparation of thiazole derivatives Dow AgroSciences LLC (US) 2013-06-19 EP disclosed
EP-2604268-A1 Process for the preparation of thiazole derivatives Dow AgroSciences LLC (US) 2013-06-19 EP disclosed
US-20130089622-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2013-04-11 US disclosed
US-20130089622-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2013-04-11 US disclosed
US-20130072382-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2013-03-21 US disclosed
US-20130072382-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2013-03-21 US disclosed
US-8350044-B2 Pesticidal compositions DOW AGROSCIENCES, LLC. (US) 2013-01-08 US disclosed
US-8350044-B2 Pesticidal compositions DOW AGROSCIENCES, LLC. (US) 2013-01-08 US disclosed
US-20100292253-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2010-11-18 US disclosed
US-20100292253-A1 PESTICIDAL COMPOSITIONS DOW AGROSCIENCES LLC (US) 2010-11-18 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100292253-A1 PESTICIDAL COMPOSITIONS ACHE, DDT, PRDX6 PIK3CG 795/4885DYRK1A 3841/4885TBK1 3723/4885
US-20130089622-A1 PESTICIDAL COMPOSITIONS ACHE, DDT, PRDX6 PIK3CG 795/4885DYRK1A 3841/4885TBK1 3723/4885
US-20150045218-A1 PESTICIDAL COMPOSITIONS ACHE, DDT, PRDX6 PIK3CG 795/4885DYRK1A 3841/4885TBK1 3723/4885
US-20130072382-A1 PESTICIDAL COMPOSITIONS ACHE, DDT, PRDX6 PIK3CG 795/4885DYRK1A 3841/4885TBK1 3723/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.