SCHEMBL13060643

SCHEMBL13060643

CCc1cccc(-c2cccc(C(=O)N[C@H](Cc3ccccc3)CN(C)C)c2)c1OC

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.44
ROCK1 Q13464 4/20 0.44
HDAC4 P56524 4/20 0.44
HDAC6 Q9UBN7 4/20 0.44
ALDH1A1 P00352 1/20 0.43
MME P08473 1/20 0.43
MMEL1 Q495T6 1/20 0.43
GPR139 Q6DWJ6 1/20 0.41
CTSL P07711 1/20 0.41
HPGDS O60760 1/20 0.41
CTRB1 P17538 1/20 0.41
HDAC1 Q13547 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13061226 1.00 ROCK2 (0.44) ROCK2ROCK1HDAC4HDAC6ALDH1A1
SCHEMBL13005496 0.93 MME (0.43) ROCK2ROCK1HDAC4HDAC6ALDH1A1
SCHEMBL13005524 0.93 MME (0.43) ROCK2ROCK1HDAC4HDAC6ALDH1A1
SCHEMBL13005652 0.87 TAS1R3 (0.43) ALDH1A1MMEMMEL1GPR139CTRB1
SCHEMBL13005647 0.87 TAS1R3 (0.43) ALDH1A1MMEMMEL1GPR139CTRB1
SCHEMBL13060890 0.87 CTSL (0.41) ROCK2ROCK1HDAC4CTSL
SCHEMBL13060892 0.87 CTSL (0.41) ROCK2ROCK1HDAC4CTSL
SCHEMBL13060640 0.86 TAS1R3 (0.40) ROCK2ROCK1CTSL
SCHEMBL13061023 0.85 ROCK2 (0.51) ROCK2ROCK1
SCHEMBL13257487 0.83 BACE1 (0.42) ROCK2ROCK1HDAC4HDAC6ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed