SCHEMBL13060640

SCHEMBL13060640

CCc1cccc(-c2cccc(C(=O)N[C@H](CN(C)C)CC(C)(C)C)c2)c1OC

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TAS1R3 Q7RTX0 4/20 0.40
TAS1R1 Q7RTX1 4/20 0.40
ROCK2 O75116 2/20 0.39
ROCK1 Q13464 2/20 0.39
UTS2R Q9UKP6 6/20 0.38
CTSL P07711 1/20 0.37
CTSS P25774 1/20 0.37
CTSK P43235 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13005620 0.92 ROCK2 (0.38) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13005639 0.92 ROCK2 (0.38) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13060892 0.87 CTSL (0.41) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13060890 0.87 CTSL (0.41) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13061226 0.86 ROCK2 (0.44) ROCK2ROCK1CTSL
SCHEMBL13060643 0.86 ROCK2 (0.44) ROCK2ROCK1CTSL
SCHEMBL13061114 0.83 TAS1R3 (0.41) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13060800 0.83 TAS1R3 (0.41) TAS1R3TAS1R1ROCK2ROCK1UTS2R
SCHEMBL13060644 0.83 CTSS (0.44) TAS1R3TAS1R1ROCK2ROCK1CTSL
SCHEMBL13060805 0.83 CTSS (0.44) TAS1R3TAS1R1ROCK2ROCK1CTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7851637-B2 Compounds and methods for inhibiting the interaction of BCL proteins with binding partners INFINITY PHARMACEUTICALS, INC. (US) 2010-12-14 US disclosed