SCHEMBL13064448

SCHEMBL13064448

CNC[C@@H]1CCc2[nH]c3ccccc3c2[C@@H]1C

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.43
SIGMAR1 Q99720 4/20 0.40
NR2E1 Q9Y466 1/20 0.40
KMT2A Q03164 1/20 0.39
DRD2 P14416 1/20 0.38
DRD1 P21728 1/20 0.38
TP53 P04637 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
RB1 P06400 2/20 0.38
SLC2A1 P11166 1/20 0.38
SLC6A4 P31645 1/20 0.37
CASP1 P29466 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24727249 0.75 SIGMAR1 (0.49) MCHR1SIGMAR1NR2E1KMT2ADRD2
SCHEMBL10748529 0.71 KDM4E (0.48) MCHR1DRD2
SCHEMBL10748537 0.71 MCHR1 (0.38) MCHR1SIGMAR1NR2E1KMT2ATP53
SCHEMBL8582769 0.69 SIGMAR1 (0.47) MCHR1SIGMAR1NR2E1KMT2ADRD2
SCHEMBL8822945 0.69 RB1 (0.45) SIGMAR1DRD2DRD1RB1
SCHEMBL19138976 0.69 KDM4E (0.40) SIGMAR1NR2E1DRD2DRD1HPGD
SCHEMBL19161133 0.69 KDM4E (0.40) SIGMAR1NR2E1DRD2DRD1HPGD
SCHEMBL17520540 0.69 KDM4E (0.40) SIGMAR1NR2E1DRD2DRD1HPGD
SCHEMBL8791963 0.67 RB1 (0.49) SIGMAR1NR2E1DRD2DRD1RB1
Hydrochloric Acid SCHEMBL8793905 0.66 RB1 (0.50) SIGMAR1NR2E1DRD2DRD1RB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010134846-A1 SUBSTITUTED 8-SULFONYL-2,3,4,5-TETRAHYDRO-1H-GAMMA-CARBOLINES, LIGANDS AND PHARMACEUTICAL COMPOSITION; METHOD FOR THE PRODUCTION AND USE OF SAME IVASHCHENKO ANDREY ALEXANDROVICH (RU) 2010-11-25 WO disclosed