SCHEMBL13070899

SCHEMBL13070899

COc1cc(/C=C/C(=O)NCCNC(=O)OC(C)(C)C)ccc1C=O

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TYR P14679 2/20 0.54
LY96 Q9Y6Y9 1/20 0.53
KDM4E B2RXH2 4/20 0.52
ALDH1A1 P00352 4/20 0.52
PKM P14618 2/20 0.52
POLB P06746 1/20 0.52
ACHE P22303 1/20 0.48
HPGD P15428 1/20 0.47
TRPV1 Q8NER1 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.46
MAOA P21397 1/20 0.46
MAOB P27338 1/20 0.46
ALOX5 P09917 2/20 0.45
MAPT P10636 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13003000 0.89 KDM4E (0.65) TYRKDM4EALDH1A1PKMPOLB
SCHEMBL1064874 0.80 KMT2A (0.51) KDM4EALDH1A1PKMHPGDSMN1; SMN2
SCHEMBL1064876 0.80 KMT2A (0.51) KDM4EALDH1A1PKMHPGDSMN1; SMN2
SCHEMBL1341952 0.78 PYGL (0.73) ALDH1A1HPGD
SCHEMBL1344394 0.78 PYGL (0.73) ALDH1A1HPGD
SCHEMBL2636844 0.77 KDM4E (0.46) KDM4EALDH1A1TRPV1SMN1; SMN2MAPT
SCHEMBL2636843 0.77 KDM4E (0.46) KDM4EALDH1A1TRPV1SMN1; SMN2MAPT
SCHEMBL18544361 0.76 CA12 (0.53) LY96KDM4EALDH1A1MAOBMAPT
SCHEMBL20085745 0.75 TOP2A (0.66)
SCHEMBL18569800 0.75 NFE2L2 (0.61) TYRKDM4EALDH1A1PKMPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2253621-A1 A SET OF GELDANAMYCIN DERIVATIVES AND THEIR PREPARATION METHODS Institute Of Medicinal Biotechnology, Chinese Academy of Medical Sciences (CN) 2010-11-24 EP disclosed