SCHEMBL13071408

SCHEMBL13071408

CC1(S(=O)(=O)NC(=O)[C@H]2C[C@H]2/C=C\CCCCC[C@H](Nc2cc(F)cc(C(F)(F)F)c2)C(=O)N2CCC[C@H]2C(N)=O)CC1

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
XIAP P98170 4/20 0.33
UBE2M P61081 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31
DPP4 P27487 1/20 0.31
F2R P25116 1/20 0.30
S1PR2 O95136 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13071891 0.94 XIAP (0.33) XIAPUBE2MDCUN1D1S1PR2
SCHEMBL13071885 0.91 XIAP (0.35) XIAPDPP4
SCHEMBL13071626 0.91 DPP4 (0.36) XIAPDPP4
SCHEMBL13071393 0.90 DPP4 (0.32) XIAPUBE2MDCUN1D1DPP4F2R
SCHEMBL13071403 0.89 USP2 (0.34) F2R
SCHEMBL12831783 0.88 F2R (0.34) XIAPF2R
SCHEMBL13072075 0.88 XIAP (0.31) XIAP
SCHEMBL13071921 0.87 DPP4 (0.35) XIAPUBE2MDCUN1D1DPP4F2R
SCHEMBL12831720 0.86 ACE (0.37)
SCHEMBL13071880 0.86 UBE2M (0.34) XIAPUBE2MDCUN1D1DPP4F2R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009142842-A9 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2010-11-25 WO disclosed
WO-2009142842-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2009-11-26 WO disclosed