SCHEMBL13071880

SCHEMBL13071880

CCOC(=O)[C@H]1C[C@H]1/C=C\CCCCC[C@H](Nc1cc(F)cc(C(F)(F)F)c1)C(=O)N1CCC[C@H]1C(N)=O

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
UBE2M P61081 4/20 0.34
DCUN1D1 Q96GG9 4/20 0.34
DPP4 P27487 1/20 0.33
XIAP P98170 2/20 0.32
F2R P25116 2/20 0.32
ALDH1A1 P00352 2/20 0.31
ACE P12821 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CXCR3 P49682 1/20 0.31
KDM4E B2RXH2 1/20 0.31
TACR2 P21452 1/20 0.31
TACR1 P25103 1/20 0.31
S1PR2 O95136 1/20 0.31
TRHR P34981 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13071404 0.91 ALDH1A1 (0.39) UBE2MDCUN1D1DPP4XIAPALDH1A1
SCHEMBL13071527 0.90 DPP4 (0.39) DPP4XIAPALDH1A1ACESMN1; SMN2
SCHEMBL13071921 0.90 DPP4 (0.35) UBE2MDCUN1D1DPP4XIAPF2R
SCHEMBL13072076 0.89 ACE (0.35) F2RALDH1A1ACESMN1; SMN2TACR1
SCHEMBL13071528 0.88 DPP4 (0.36) DPP4F2RACESMN1; SMN2
SCHEMBL13071526 0.87 UBE2M (0.35) UBE2MDCUN1D1XIAPF2RACE
SCHEMBL13071393 0.87 DPP4 (0.32) UBE2MDCUN1D1DPP4XIAPF2R
SCHEMBL13071408 0.86 XIAP (0.33) UBE2MDCUN1D1DPP4XIAPF2R
SCHEMBL12831754 0.85 ACE (0.41) ACESMN1; SMN2
SCHEMBL13071891 0.80 XIAP (0.33) UBE2MDCUN1D1XIAPS1PR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009142842-A9 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2010-11-25 WO disclosed
WO-2009142842-A2 NOVEL MACROCYCLIC INHIBITORS OF HEPATITIS C VIRUS REPLICATION INTERMUNE, INC. (US) 2009-11-26 WO disclosed