SCHEMBL1307300

SCHEMBL1307300

O=C(c1ccc(-c2ccco2)cc1F)c1c(F)c(F)c(F)c(F)c1F

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.45
KAT6A Q92794 3/20 0.44
KEAP1 Q14145 1/20 0.43
USP2 O75604 2/20 0.40
POLB P06746 2/20 0.40
NR4A2 P43354 1/20 0.38
PTPN1 P18031 1/20 0.38
HDAC2 Q92769 1/20 0.38
PGR P06401 1/20 0.38
TDP2 O95551 2/20 0.37
ATM Q13315 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PPARG P37231 1/20 0.37
PPARA Q07869 1/20 0.37
GPR17 Q13304 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
ALDH1A1 P00352 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1309155 0.80 TUBB4A (0.47) ERN1KAT6ANR4A2ALDH1A1
SCHEMBL1308192 0.76 TUBB4A (0.38) ERN1KAT6AKEAP1POLBNR4A2
SCHEMBL12113575 0.75 TUBB4A (0.66) ALDH1A1
SCHEMBL28269364 0.72 ERN1 (0.54) ERN1KAT6AKEAP1USP2POLB
SCHEMBL22126675 0.68 HNF4A (0.59) ERN1KEAP1POLBPTPN1L3MBTL1
SCHEMBL19155098 0.68 ERN1 (0.47) ERN1KAT6AKEAP1USP2POLB
SCHEMBL6521942 0.67 KEAP1 (0.47) ERN1KAT6AKEAP1USP2POLB
SCHEMBL27623999 0.66 TAAR1 (0.55) ERN1KEAP1USP2POLBHDAC2
SCHEMBL20462888 0.65 ERN1 (0.46) ERN1KAT6AKEAP1PGRTAAR1
SCHEMBL27605185 0.65 KEAP1 (0.77) ERN1KAT6AKEAP1USP2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8053439-B2 Benzophenone derivatives useful for inhibiting formation of microtubule CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2011-11-08 US claimed
US-20090275575-A1 BENZOPHENONE DERIVATIVES USEFUL FOR INHIBITING FORMATION OF MICROTUBULE CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2009-11-05 US claimed
EP-2066632-A1 BENZOPHENONE DERIVATIVES USEFUL FOR INHIBITING FORMATION OF MICROTUBULE Chong Kun Dang Pharmaceutical Corp. (KR) 2009-06-10 EP claimed
WO-2008038955-A1 BENZOPHENONE DERIVATIVES USEFUL FOR INHIBITING FORMATION OF MICROTUBULE CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2008-04-03 WO claimed
EP-2066632-B1 BENZOPHENONE DERIVATIVES USEFUL FOR INHIBITING FORMATION OF MICROTUBULE CHONG KUN DANG PHARM CORP (KR) 2013-09-04 EP disclosed
US-8053439-B2 Benzophenone derivatives useful for inhibiting formation of microtubule CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2011-11-08 US disclosed
US-8053439-B2 Benzophenone derivatives useful for inhibiting formation of microtubule CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2011-11-08 US disclosed
US-8053439-B2 Benzophenone derivatives useful for inhibiting formation of microtubule CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2011-11-08 US disclosed
US-20090275575-A1 BENZOPHENONE DERIVATIVES USEFUL FOR INHIBITING FORMATION OF MICROTUBULE CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2009-11-05 US disclosed
US-20090275575-A1 BENZOPHENONE DERIVATIVES USEFUL FOR INHIBITING FORMATION OF MICROTUBULE CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2009-11-05 US disclosed
US-20090275575-A1 BENZOPHENONE DERIVATIVES USEFUL FOR INHIBITING FORMATION OF MICROTUBULE CHONG KUN DANG PHARMACEUTICAL CORP. (KR) 2009-11-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090275575-A1 BENZOPHENONE DERIVATIVES USEFUL FOR INHIBITING FORMATION OF MICROTUBULE TUBB1, TUBA1C, TUBB6 ERN1 2333/4885KAT6A 493/4885KEAP1 1140/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.