SCHEMBL13076252

SCHEMBL13076252

Fc1cccc(Cl)c1-c1nc(-c2ccc(-c3ccc(OC(F)(F)F)cc3)nc2)c(Br)[nH]1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGES O14684 16/20 0.57
PTGS1 P23219 2/20 0.48
MAPK14 Q16539 2/20 0.38
NR3C1 P04150 1/20 0.36
JAK2 O60674 1/20 0.36
CBFB Q13951 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13076280 0.92 PTGES (0.56) PTGESPTGS1MAPK14
SCHEMBL3799807 0.86 PTGES (0.43) PTGESPTGS1MAPK14JAK2CBFB
SCHEMBL3791947 0.84 PTGES (0.61) PTGESPTGS1MAPK14JAK2
SCHEMBL13075522 0.83 PTGES (0.65) PTGESPTGS1MAPK14
SCHEMBL13075554 0.82 PTGES (0.64) PTGESMAPK14JAK2
SCHEMBL13075547 0.80 PTGES (0.56) PTGESPTGS1MAPK14JAK2
SCHEMBL3798464 0.79 PTGES (0.50) PTGESPTGS1MAPK14
SCHEMBL13076254 0.79 PTGES (0.54) PTGESPTGS1MAPK14
SCHEMBL13075515 0.78 PTGES (0.64) PTGESPTGS1MAPK14
SCHEMBL13076241 0.77 PTGES (0.55) PTGESPTGS1MAPK14JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed