SCHEMBL3799807

SCHEMBL3799807

Fc1cccc(Cl)c1-c1nc(Br)c(-c2ccc(-c3ccc(OC(F)(F)F)cc3)nc2)[nH]1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGES O14684 16/20 0.43
PTGS1 P23219 1/20 0.42
MAPK14 Q16539 2/20 0.38
JAK2 O60674 1/20 0.36
DGAT1 O75907 1/20 0.35
CBFB Q13951 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3798464 0.92 PTGES (0.50) PTGESPTGS1MAPK14DGAT1CYP2C9
SCHEMBL13076252 0.86 PTGES (0.57) PTGESPTGS1MAPK14JAK2CBFB
SCHEMBL3805843 0.84 PTGES (0.46) PTGESMAPK14JAK2CYP2C9
SCHEMBL3790737 0.83 PTGES (0.49) PTGESPTGS1MAPK14CYP2C9
SCHEMBL3793065 0.82 PTGES (0.47) PTGESMAPK14JAK2CYP2C9
SCHEMBL3796330 0.80 PTGES (0.41) PTGESMAPK14JAK2CYP2C9
SCHEMBL13076280 0.79 PTGES (0.56) PTGESPTGS1MAPK14
SCHEMBL3795197 0.78 PTGES (0.47) PTGESMAPK14JAK2CYP2C9
SCHEMBL3799359 0.77 PTGES (0.44) PTGESMAPK14CYP2C9
SCHEMBL3795498 0.76 PTGES (0.45) PTGESMAPK14JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO claimed
WO-2010127152-A2 COMPOUNDS AND COMPOSITIONS AS MICROSOMAL PROSTAGLANDIN E SYNTHASE-1 INHIBITORS IRM LLC (BM) 2010-11-04 WO disclosed