SCHEMBL1309845

SCHEMBL1309845

O=c1[nH]c(=O)c2oc3ccccc3c2[nH]1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 1/20 0.54
FEN1 P39748 1/20 0.54
ALDH1A1 P00352 7/20 0.51
KDM4E B2RXH2 6/20 0.51
LMNA P02545 4/20 0.51
GLA P06280 3/20 0.51
HSD17B10 Q99714 2/20 0.51
GAA P10253 1/20 0.51
TSHR P16473 1/20 0.51
RXFP1 Q9HBX9 7/20 0.50
PPARG P37231 6/20 0.50
NR2E3 Q9Y5X4 6/20 0.50
NCOR2 Q9Y618 6/20 0.50
HTT P42858 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
NPSR1 Q6W5P4 3/20 0.46
MAPT P10636 3/20 0.45
KMT2A Q03164 2/20 0.45
MEN1 O00255 1/20 0.45
CSF1R P07333 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5323077 0.80 ALDH1A1 (0.56) ERCC5FEN1ALDH1A1KDM4ELMNA
SCHEMBL18774623 0.78 ERCC5 (0.56) ERCC5FEN1ALDH1A1KDM4ELMNA
SCHEMBL24665384 0.78 ERCC5 (0.49) ERCC5FEN1ALDH1A1KDM4ELMNA
SCHEMBL2497885 0.77 PIM1 (0.54) ALDH1A1LMNAHSD17B10TSHRRXFP1
SCHEMBL22006946 0.77 DAO (0.46) ALDH1A1LMNAHSD17B10TSHRRXFP1
SCHEMBL30914138 0.77 MAOB (0.40) ALDH1A1KDM4ELMNARXFP1PPARG
SCHEMBL1854409 0.77 PIM1 (0.54) PIM1CSNK2A2CSNK2BPIM3PIM2
SCHEMBL8691721 0.75 ERCC5 (0.54) ERCC5FEN1ALDH1A1KDM4ELMNA
SCHEMBL22006356 0.75 PIM1 (0.41) CA12PARP1CA9PIM1CSNK2A2
SCHEMBL22006833 0.75 AHR (0.42) KDM4ECSF1RPDGFRBCA12PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 24 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4615578-A1 CYCLIC PYRIDINE DERIVATIVES AS CGAS INHIBITORS Boehringer Ingelheim International GmbH (DE) 2025-09-17 EP disclosed
EP-4615849-A1 CYCLIC BENZIMIDAZOLE DERIVATIVES AS CGAS INHIBITORS Boehringer Ingelheim International GmbH (DE) 2025-09-17 EP disclosed
CN-120202206-A Cyclic benzimidazole derivatives as cGAS inhibitors 勃林格殷格翰国际有限公司 2025-06-24 CN disclosed
US-20240208997-A1 CYCLIC BENZIMIDAZOLE DERIVATIVES AS CGAS INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2024-06-27 US disclosed
US-20240208997-A1 CYCLIC BENZIMIDAZOLE DERIVATIVES AS CGAS INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2024-06-27 US disclosed
US-20240189315-A1 Cyclic Pyridine Derivatives as cGAS Inhibitors BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2024-06-13 US disclosed
WO-2024099907-A1 CYCLIC BENZIMIDAZOLE DERIVATIVES AS CGAS INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2024-05-16 WO disclosed
WO-2024099908-A1 CYCLIC PYRIDINE DERIVATIVES AS CGAS INHIBITORS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2024-05-16 WO disclosed
US-10361377-B2 Condensed cyclic compound and organic light emitting device including the same SAMSUNG SDI CO., LTD. (KR) 2019-07-23 US disclosed
US-20160308142-A1 CONDENSED CYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME SAMSUNG ELECTRONICS CO., LTD. (KR) 2016-10-20 US disclosed
WO-2015105315-A1 FUSED-RING COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE COMPRISING SAME 삼성에스디아이 주식회사 2015-07-16 WO disclosed
US-8921361-B2 Triazine, pyrimidine and pyridine analogs and their use as therapeutic agents and diagnostic probes UNIVERSITY OF BASEL (CH) 2014-12-30 US disclosed
US-8921361-B2 Triazine, pyrimidine and pyridine analogs and their use as therapeutic agents and diagnostic probes UNIVERSITY OF BASEL (CH) 2014-12-30 US disclosed
US-8921361-B2 Triazine, pyrimidine and pyridine analogs and their use as therapeutic agents and diagnostic probes UNIVERSITY OF BASEL (CH) 2014-12-30 US disclosed
US-20110275762-A1 TRIAZINE, PYRIMIDINE AND PYRIDINE ANALOGS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES UNIVERSITY OF BASEL (CH) 2011-11-10 US disclosed
US-20110275762-A1 TRIAZINE, PYRIMIDINE AND PYRIDINE ANALOGS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES UNIVERSITY OF BASEL (CH) 2011-11-10 US disclosed
US-20110275762-A1 TRIAZINE, PYRIMIDINE AND PYRIDINE ANALOGS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES UNIVERSITY OF BASEL (CH) 2011-11-10 US disclosed
EP-2364302-A2 TRIAZINE, PYRIMIDINE AND PYRIDINE ANALOGS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES University of Basel (CH) 2011-09-14 EP disclosed
WO-2010052569-A2 TRIAZINE, PYRIMIDINE AND PYRIDINE ANALOGS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES UNIVERSITY OF BASEL (CH) 2010-05-14 WO disclosed
WO-2010052569-A2 TRIAZINE, PYRIMIDINE AND PYRIDINE ANALOGS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES UNIVERSITY OF BASEL (CH) 2010-05-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110275762-A1 TRIAZINE, PYRIMIDINE AND PYRIDINE ANALOGS AND THEIR USE AS THERAPEUTIC AGENTS AND DIAGNOSTIC PROBES MTOR, PIK3CA, PIK3CD ERCC5 3213/4885FEN1 3147/4885ALDH1A1 3410/4885
US-20160308142-A1 CONDENSED CYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME CRY1, CRY2, CCNE2 ERCC5 133/4885FEN1 1993/4885ALDH1A1 1905/4885
US-20240208997-A1 CYCLIC BENZIMIDAZOLE DERIVATIVES AS CGAS INHIBITORS CGAS, STING1, IFNAR1 ERCC5 2747/4885FEN1 490/4885ALDH1A1 815/4885
US-20240189315-A1 Cyclic Pyridine Derivatives as cGAS Inhibitors CGAS, STING1, IRF3 ERCC5 2719/4885FEN1 229/4885ALDH1A1 1257/4885
US-10361377-B2 Condensed cyclic compound and organic light emitting device including the same CRY1, CRY2, CCNE2 ERCC5 122/4885FEN1 2034/4885ALDH1A1 1077/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.