SCHEMBL13115682

SCHEMBL13115682

CCOC(=O)Cn1cnc2ccn(-c3ccc(C)cc3)c(=O)c21

nearest known ligand 0.57

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.57
LMNA P02545 1/20 0.57
GAA P10253 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
RAB9A P51151 3/20 0.47
HTT P42858 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 2/20 0.47
KMT2A Q03164 2/20 0.47
MAPT P10636 1/20 0.47
HSD17B10 Q99714 1/20 0.47
CYP2C19 P33261 1/20 0.46
NPC1 O15118 1/20 0.46
POLB P06746 2/20 0.45
KDM4E B2RXH2 1/20 0.44
USP2 O75604 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13115679 0.86 ADORA2B (0.46) TSHRLMNAGAARAB9AHTT
SCHEMBL18956047 0.82 RAB9A (0.60) TSHRLMNAGAAL3MBTL1RAB9A
SCHEMBL13575231 0.82 LMNA (0.48) TSHRLMNAGAAL3MBTL1RAB9A
SCHEMBL13115685 0.72 LMNA (0.46) TSHRLMNAGAAL3MBTL1RAB9A
SCHEMBL3594719 0.72 RXFP1 (0.42) LMNARAB9AHTTALDH1A1KMT2A
SCHEMBL14564343 0.70 ALDH1A1 (0.49) TSHRLMNAL3MBTL1RAB9AHTT
SCHEMBL28149945 0.69 RAB9A (0.65) TSHRLMNARAB9AALDH1A1KMT2A
SCHEMBL12260494 0.69 SMN1; SMN2 (0.76) TSHRLMNAL3MBTL1MEN1KMT2A
SCHEMBL7404412 0.67 ALDH1A1 (0.65) TSHRLMNAL3MBTL1HTTALDH1A1
SCHEMBL659913 0.67 TSHR (0.52) TSHRLMNAGAAL3MBTL1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7807704-B2 Bicyclic, nitrogen-containing compounds modulating CXCR4 and/or CCXCKR2 CHEMOCENTRYX, INC. (US) 2010-10-05 US disclosed
US-7807704-B2 Bicyclic, nitrogen-containing compounds modulating CXCR4 and/or CCXCKR2 CHEMOCENTRYX, INC. (US) 2010-10-05 US disclosed
US-20070275965-A1 CXCR4 modulators CHEMOCENTRYX, INC. (US) 2007-11-29 US disclosed
US-20070275965-A1 CXCR4 modulators CHEMOCENTRYX, INC. (US) 2007-11-29 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070275965-A1 CXCR4 modulators CXCL12, CXCR4, CXCR1 TSHR 1277/4885LMNA 4638/4885GAA 1982/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.