SCHEMBL13147677

SCHEMBL13147677

Cc1nn(C)c(C)c1-c1cc(N)nc(-c2nc(C(F)(F)F)cs2)n1

nearest known ligand 0.37

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
GAA P10253 2/20 0.37
ABL1 P00519 1/20 0.36
BCR P11274 1/20 0.36
MAP4K1 Q92918 2/20 0.35
IDH1 O75874 4/20 0.34
GPBAR1 Q8TDU6 1/20 0.34
KDM4E B2RXH2 4/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MCHR1 Q99705 1/20 0.33
LMNA P02545 2/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
PRMT6 Q96LA8 1/20 0.32
HPGD P15428 3/20 0.31
TGFBR1 P36897 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL585936 0.88 ABL1 (0.36) ALDH1A1GAAABL1BCRMAP4K1
SCHEMBL586384 0.80 ABL1 (0.34) ALDH1A1GAAABL1BCRIDH1
SCHEMBL13147740 0.79 IDH1 (0.41) ALDH1A1IDH1KDM4ETGFBR1
SCHEMBL13147681 0.79 IDH1 (0.36) ALDH1A1IDH1GPBAR1NPC1RAB9A
SCHEMBL13147680 0.77 PTGS2 (0.40) IDH1LMNAMAPT
SCHEMBL13147664 0.77 ALDH1A1 (0.44) ALDH1A1IDH1KDM4ELMNANPC1
SCHEMBL13147748 0.77 IDH1 (0.36) ALDH1A1IDH1NPC1PRMT6MAPT
SCHEMBL13147745 0.76 IDH1 (0.38) ALDH1A1IDH1KDM4ELMNAHPGD
SCHEMBL586224 0.76 ABL1 (0.37) GAAABL1BCRL3MBTL1MCHR1
SCHEMBL13147682 0.76 LMNA (0.45) ALDH1A1GAAIDH1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118078-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed