SCHEMBL13147682

SCHEMBL13147682

Cc1nc(C)c(-c2cc(N)nc(-c3nc(C(F)(F)F)cs3)n2)s1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.45
HTT P42858 1/20 0.45
OPRM1 P35372 5/20 0.40
CDK2 P24941 2/20 0.39
CDK4 P11802 1/20 0.39
CCNE1 P24864 1/20 0.39
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
NPC1 O15118 3/20 0.38
GAA P10253 1/20 0.38
RAB9A P51151 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
GFER P55789 1/20 0.36
IDH1 O75874 3/20 0.35
TRPV4 Q9HBA0 3/20 0.35
COMT P21964 1/20 0.34
TUBB4A P04350 1/20 0.34
TUBB P07437 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL578009 0.87 OPRM1 (0.40) LMNAHTTOPRM1CDK2CDK4
SCHEMBL3072583 0.83 OPRM1 (0.38) LMNAHTTOPRM1CDK2MEN1
SCHEMBL13147664 0.83 ALDH1A1 (0.44) LMNAHTTKMT2ANPC1RAB9A
SCHEMBL13147670 0.82 KDM4E (0.36) HTTMEN1KMT2AKDM4EALDH1A1
SCHEMBL13147748 0.82 IDH1 (0.36) NPC1ALDH1A1MAPTGFERIDH1
SCHEMBL13147740 0.82 IDH1 (0.41) KMT2AKDM4EALDH1A1IDH1
SCHEMBL13147680 0.80 PTGS2 (0.40) LMNACDK2MAPTIDH1
SCHEMBL13147658 0.80 IDH1 (0.36) NPC1KDM4EALDH1A1MAPTGFER
SCHEMBL13147672 0.79 SRC (0.38) CDK2NPC1ALDH1A1MAPTGFER
SCHEMBL578105 0.79 LMNA (0.39) LMNAHTTOPRM1CDK2CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118078-A1 MACROCYCLIC SERINE PROTEASE INHIBITORS IDENIX PHARMACEUTICALS, INC. (US) 2010-10-14 WO disclosed