SCHEMBL1316360

SCHEMBL1316360

COc1ccc(C(=O)NCc2cccc(-c3ccco3)c2)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.58
RAB9A P51151 3/20 0.58
CHRM3 P20309 1/20 0.58
ALDH1A1 P00352 4/20 0.57
MMP13 P45452 3/20 0.56
ROCK2 O75116 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
PRKACA P17612 1/20 0.55
GSK3A P49840 1/20 0.55
GSK3B P49841 1/20 0.55
PRKX P51817 1/20 0.55
PRKCQ Q04759 1/20 0.55
ROCK1 Q13464 1/20 0.55
CLK4 Q9HAZ1 1/20 0.55
PRMT6 Q96LA8 1/20 0.54
ADORA2A P29274 2/20 0.53
ADORA1 P30542 2/20 0.53
ADORA3 P0DMS8 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1319516 0.90 MMP13 (0.66) NPC1RAB9ACHRM3ALDH1A1MMP13
SCHEMBL1317763 0.87 TDP1 (0.59) NPC1RAB9AALDH1A1MMP13CYP3A4
SCHEMBL1317036 0.84 PRMT6 (0.54) NPC1RAB9ACHRM3ALDH1A1ROCK2
SCHEMBL1315943 0.84 PRMT6 (0.54) NPC1RAB9AALDH1A1MMP13ROCK2
SCHEMBL15428870 0.83 KMT2A (0.67) NPC1RAB9ACHRM3ALDH1A1MMP13
SCHEMBL1316394 0.83 KMT2A (0.61) NPC1RAB9AALDH1A1PRMT6ADORA2A
SCHEMBL1317297 0.82 CHRM3 (0.59) NPC1RAB9ACHRM3ALDH1A1ROCK2
SCHEMBL1318282 0.81 POLB (0.64) NPC1RAB9ACHRM3ALDH1A1PRMT6
SCHEMBL1317667 0.79 PRMT6 (0.53) NPC1RAB9AALDH1A1MMP13ROCK2
SCHEMBL1317689 0.79 CHRM3 (0.58) CHRM3ALDH1A1ROCK2ROCK1PRMT6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8637550-B2 Heteroaryl diamide compounds useful as MMP-13 inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2014-01-28 US disclosed
US-20110275625-A1 Heteroaryl Diamide Compounds Useful as MMP-13 Inhibitors BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-11-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110275625-A1 Heteroaryl Diamide Compounds Useful as MMP-13 Inhibitors MMP13, MMP3, MMP11 NPC1 1853/4885RAB9A 1137/4885CHRM3 4240/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.