SCHEMBL13178294

SCHEMBL13178294

O=C(c1ccc(I)cc1)C(Br)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.60
CES2 O00748 3/20 0.53
CES1 P23141 3/20 0.53
PDPK1 O15530 2/20 0.53
TDP1 Q9NUW8 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
TPMT P51580 1/20 0.47
LMNA P02545 3/20 0.46
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
ALDH1A1 P00352 2/20 0.40
HSD17B10 Q99714 1/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.38
SRC P12931 1/20 0.38
ADORA3 P0DMS8 1/20 0.37
PTPN1 P18031 1/20 0.37
PTPN6 P29350 1/20 0.37
PTPN11 Q06124 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL627867 0.86 CES2 (0.64) CES2CES1TDP1L3MBTL1LMNA
SCHEMBL5525568 0.83 CES2 (0.55) CES2CES1TDP1L3MBTL1LMNA
SCHEMBL2976217 0.83 LMNA (0.57) CES2CES1PDPK1TDP1L3MBTL1
SCHEMBL5318489 0.82 GSK3B (0.56) GSK3BCES2CES1PDPK1TPMT
SCHEMBL682581 0.81 CES2 (0.53) CES2CES1TDP1L3MBTL1LMNA
SCHEMBL627839 0.81 CES2 (0.53) CES2CES1PDPK1TDP1L3MBTL1
SCHEMBL10824473 0.80 CES2 (0.52) CES2CES1TDP1L3MBTL1LMNA
SCHEMBL28878867 0.79 ALDH1A1 (0.53) CES2CES1TDP1L3MBTL1LMNA
SCHEMBL16682291 0.79 CES2 (0.50) CES2CES1PDPK1TDP1L3MBTL1
SCHEMBL1429237 0.79 ALDH1A1 (0.50) CES2CES1TDP1L3MBTL1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501819-B1 ESTROGEN RECEPTOR MODULATORS MERCK SHARP & DOHME (US) 2010-09-15 EP disclosed