SCHEMBL13186597

SCHEMBL13186597

C/C=C1\NCCc2cc(C(C)=O)ccc21

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
MAPT P10636 1/20 0.51
PARP10 Q53GL7 3/20 0.51
PARP11 Q9NR21 3/20 0.51
HSD17B1 P14061 1/20 0.45
KMT2A Q03164 4/20 0.43
MEN1 O00255 2/20 0.43
KCNJ1 P48048 1/20 0.39
PRKACA P17612 1/20 0.37
PRKACG P22612 1/20 0.37
PRKACB P22694 1/20 0.37
S100A4 P26447 1/20 0.37
PGR P06401 1/20 0.37
SRD5A1 P18405 3/20 0.36
SRD5A2 P31213 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1727165 0.81 PARP11 (0.72) NPC1RAB9AMAPTPARP10PARP11
SCHEMBL15106295 0.76 RAB9A (0.77) NPC1RAB9AMAPTPARP10PARP11
SCHEMBL2610325 0.76 MAPT (0.58) NPC1RAB9AMAPTPARP10PARP11
SCHEMBL13186574 0.74 PARP10 (0.47) PARP10PARP11SRD5A1
SCHEMBL11808846 0.72 MAPT (0.50) NPC1RAB9AMAPTPARP10PARP11
SCHEMBL13187114 0.72 PARP10 (0.38) MAPTPARP10PARP11KMT2AMEN1
SCHEMBL14395011 0.72 PARP10 (0.61) NPC1RAB9AMAPTPARP10PARP11
SCHEMBL1790024 0.70 NPC1 (0.56) NPC1RAB9AMAPTHSD17B1
SCHEMBL8253223 0.70 NPC1 (0.61) NPC1RAB9AMAPTPARP10PARP11
SCHEMBL29809406 0.69 SRD5A2 (0.72) NPC1RAB9AMAPTHSD17B1S100A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100070-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE F. HOFFMANN-LA ROCHE AG (CH) 2010-09-10 WO disclosed