SCHEMBL13187114

SCHEMBL13187114

C/C=C1\NCCc2cc(N(C)C)ccc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP10 Q53GL7 5/20 0.38
PARP11 Q9NR21 4/20 0.38
ALDH1A1 P00352 4/20 0.37
GAA P10253 2/20 0.35
CYP26A1 O43174 2/20 0.35
MIF P14174 1/20 0.35
ADRA2A P08913 3/20 0.34
ADRA2B P18089 2/20 0.34
ADRA2C P18825 2/20 0.34
ABCC4 O15439 1/20 0.33
ABCB11 O95342 1/20 0.33
CHRM2 P08172 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CHRM1 P11229 1/20 0.33
ACHE P22303 1/20 0.33
PTGS1 P23219 1/20 0.33
PDE4A P27815 1/20 0.33
SLC6A4 P31645 1/20 0.33
KCNH2 Q12809 1/20 0.33
PARP1 P09874 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1432600 0.79 PARP10 (0.63) PARP10PARP11PARP1GRM5
SCHEMBL13186574 0.77 PARP10 (0.47) PARP10PARP11PARP1GRM5
SCHEMBL8526314 0.74 DRD2 (0.53) ALDH1A1GAAADRA2AADRA2BADRA2C
SCHEMBL13186597 0.72 NPC1 (0.51) PARP10PARP11MEN1KMT2AMAPT
SCHEMBL5871312 0.70 GFER (0.43) PARP10ALDH1A1GAAADRA2AADRA2B
SCHEMBL2577433 0.68 HTR2C (0.53) ADRA2AADRA2BADRA2C
SCHEMBL8155747 0.68 PARP11 (0.68) PARP10PARP11PARP1GRM5
SCHEMBL6776955 0.67 CASP1 (0.53) ALDH1A1CYP26A1MIFKDM4EHSD17B10
SCHEMBL4886295 0.67 ALDH1A1 (0.46) ALDH1A1KDM4EALOX15HSD17B10LMNA
SCHEMBL3873373 0.66 PNMT (0.55) ADRA2AADRA2BADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010100070-A1 INHIBITORS OF BRUTON'S TYROSINE KINASE F. HOFFMANN-LA ROCHE AG (CH) 2010-09-10 WO disclosed