SCHEMBL13190827

SCHEMBL13190827

CC(N)c1cccc(Oc2ccc(Cl)cc2N)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.65
CYP1A2 P05177 2/20 0.60
CYP2C9 P11712 2/20 0.60
CYP2C19 P33261 2/20 0.60
CYP3A4 P08684 1/20 0.60
MAPT P10636 4/20 0.55
HTT P42858 2/20 0.55
LMNA P02545 1/20 0.55
ALDH1A1 P00352 2/20 0.54
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
KDM4E B2RXH2 1/20 0.54
CYP2D6 P10635 1/20 0.54
HPGD P15428 1/20 0.54
GAA P10253 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
ADRB2 P07550 1/20 0.40
P2RX4 Q99571 1/20 0.39
PTGER4 P35408 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2965348 0.87 L3MBTL1 (0.63) L3MBTL1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL2805226 0.81 NOS2 (0.47) L3MBTL1CYP1A2CYP2C9CYP2C19CYP3A4
Hydrochloric Acid SCHEMBL2805035 0.80 NOS2 (0.46) L3MBTL1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL2967362 0.77 MAPT (0.72) L3MBTL1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL307310 0.76 CYP1A2 (1.00) L3MBTL1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL359171 0.76 CYP1A2 (0.68) L3MBTL1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL13190865 0.76 L3MBTL1 (0.49) L3MBTL1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL811122 0.74 MAPT (0.66) L3MBTL1CYP1A2CYP2C9CYP2C19CYP3A4
SCHEMBL20511655 0.73 PTGS1 (0.62) MAPTALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL14831002 0.73 PTGS1 (0.62) MAPTALDH1A1MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010108059-A1 SUBSTITUTED PYRIMIDINE DERIVATIVES AS ANTAGONISTS OF THE HISTAMINE H4 RECEPTOR INCYTE CORPORATION (US) 2010-09-23 WO disclosed